SCHEMBL6925451

SCHEMBL6925451

CN1CCN(c2ccc(-c3nc(-c4ccccc4)c[nH]3)cn2)CC1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
FYN P06241 3/20 0.54
HRH4 Q9H3N8 3/20 0.50
HTR3A P46098 3/20 0.50
TNKS O95271 2/20 0.50
ATR Q13535 1/20 0.50
TDO2 P48775 1/20 0.48
ACVR1B P36896 1/20 0.45
TGFBR1 P36897 1/20 0.45
MET P08581 1/20 0.44
DGAT1 O75907 1/20 0.44
SOAT1 P35610 1/20 0.44
KCNH2 Q12809 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6927440 0.89 HRH4 (0.51) HRH4HTR3ATNKSTDO2DGAT1
SCHEMBL6926756 0.89 TDO2 (0.58) FYNHRH4HTR3ATNKSTDO2
SCHEMBL6925668 0.88 CNR2 (0.53) FYNATR
SCHEMBL6924524 0.87 CNR2 (0.53) FYNHRH4HTR3ATNKSTDO2
SCHEMBL6925885 0.87 CNR2 (0.56)
SCHEMBL6924723 0.87 HRH3 (0.45) FYNTNKSATRDGAT1
SCHEMBL6925622 0.87 HRH3 (0.45) FYNMET
SCHEMBL6926636 0.86 TSHR (0.46) FYNHTR3ADGAT1
SCHEMBL6924500 0.86 ATR (0.51) HTR3AATRACVR1BKCNH2
SCHEMBL6926900 0.85 CNR2 (0.53) ATRTDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6514966-B2 Neuropeptide Y antagonists such as 2-chloro-5-(4-(3,4-dich loro-phenyl)-1H-imidazol-2-yl)-pyridine PFIZER INC. 2003-02-04 US disclosed
US-6355635-B1 IMIDAZOLEBENZENE, IMIDAZOLEPYRIDINE COMPOUNDS FOR TREATMENT OF OBESITY PFIZER INC. 2002-03-12 US disclosed
US-20010039277-A1 Compounds for the treatment of obesity ELLIOTT RICHARD L (US) 2001-11-08 US disclosed
WO-2000066578-A1 COMPOUNDS FOR THE TREATMENT OF OBESITY PFIZER PRODUCTS INC. (US) 2000-11-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20010039277-A1 Compounds for the treatment of obesity NPY1R, NPY4R, NPY2R FYN 1544/4885HRH4 437/4885HTR3A 92/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.