SCHEMBL6925964

SCHEMBL6925964

C[Si](C)(C)CCOc1nc(N)nc2[nH]cnc12

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 17/20 0.43
CCNB1 P14635 17/20 0.43
CCNA2 P20248 16/20 0.43
CDK2 P24941 16/20 0.43
CCNA1 P78396 16/20 0.43
PIN1 Q13526 2/20 0.43
MGMT P16455 4/20 0.35
MPO P05164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8830293 0.85 CDK1 (0.60) CDK1CCNB1CCNA2CDK2CCNA1
SCHEMBL880169 0.84 CDK1 (0.61) CDK1CCNB1CCNA2CDK2CCNA1
SCHEMBL8537496 0.84 CDK1 (0.44) CDK1CCNB1CCNA2CDK2CCNA1
SCHEMBL12227596 0.82 CDK1 (0.42) CDK1CCNB1CCNA2CDK2CCNA1
SCHEMBL8618497 0.81 CDK1 (0.44) CDK1CCNB1CCNA2CDK2CCNA1
SCHEMBL31570032 0.80 PDPK1 (0.33) CDK1CCNB1CCNA2CDK2CCNA1
SCHEMBL13369897 0.80 PDPK1 (0.33) CDK1CCNB1CCNA2CDK2CCNA1
Methylguanine SCHEMBL29968306 0.78 CDK1 (0.41) CDK1CCNB1CCNA2CDK2CCNA1
Methylguanine SCHEMBL1336757 0.78 CDK1 (0.41) CDK1CCNB1CCNA2CDK2CCNA1
SCHEMBL821881 0.77 CDK1 (0.46) CDK1CCNB1CCNA2CDK2CCNA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040068111-A1 Unsaturated phosphonate derivatives of purines and pyrimidines AVENTIS PHARMACEUTICALS INC. 2004-04-08 US disclosed
US-20030004345-A1 Unsaturated phosphonate derivatives of purines and pyrimidines CASARA PATRICK (FR) 2003-01-02 US disclosed
EP-0701562-B1 UNSATURATED PHOSPHONATES DERIVATIVES OF PURINES AND PYRIMIDINES MERRELL PHARMA INC (US) 1997-06-18 EP disclosed
EP-0701562-A1 UNSATURATED PHOSPHONATES DERIVATIVES OF PURINES AND PYRIMIDINES MERRELL DOW PHARMA (US) 1996-03-20 EP disclosed
WO-1994022882-A1 UNSATURATED PHOSPHONATES DERIVATIVES OF PURINES AND PYRIMIDINES MERRELL DOW PHARMACEUTICALS INC. (US) 1994-10-13 WO disclosed
EP-0618214-A1 Unsaturated phosphonate derivatives of purines and pyrimidines MERRELL DOW PHARMACEUTICALS INC. (US) 1994-10-05 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040068111-A1 Unsaturated phosphonate derivatives of purines and pyrimidines TYMP, NUDT1, PNP CDK1 521/4885CCNB1 825/4885CCNA2 822/4885
US-20030004345-A1 Unsaturated phosphonate derivatives of purines and pyrimidines TYMP, NUDT1, PNP CDK1 521/4885CCNB1 825/4885CCNA2 822/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.