SCHEMBL6926258

SCHEMBL6926258

COc1ccc(C(=O)Nc2ccc(-c3ccccc3)cc2)cc1O

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCC1 P33527 2/20 0.76
ABCB1 P08183 2/20 0.65
MEN1 O00255 1/20 0.64
KMT2A Q03164 1/20 0.64
NAMPT P43490 1/20 0.61
HDAC1 Q13547 1/20 0.60
HDAC8 Q9BY41 1/20 0.60
HDAC6 Q9UBN7 1/20 0.60
PDE4D Q08499 1/20 0.59
DEGS1 O15121 1/20 0.58
PTPN1 P18031 1/20 0.58
PLAU P00749 2/20 0.57
CYP3A4 P08684 2/20 0.57
CYP1A2 P05177 1/20 0.57
POLB P06746 1/20 0.57
ALDH1A1 P00352 2/20 0.57
MAPT P10636 1/20 0.57
MCHR1 Q99705 1/20 0.57
TRPV1 Q8NER1 1/20 0.56
TSHR P16473 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30873016 0.92 MEN1 (0.70) ABCC1ABCB1MEN1KMT2ANAMPT
SCHEMBL7147243 0.92 MEN1 (0.70) ABCC1ABCB1MEN1KMT2ANAMPT
SCHEMBL3245372 0.86 NAMPT (0.65) ABCC1MEN1KMT2ANAMPTPDE4D
SCHEMBL18007344 0.85 HPSE (0.66) ABCC1MEN1KMT2AHDAC1HDAC8
SCHEMBL18007317 0.85 ABCC1 (0.63) ABCC1MEN1KMT2AHDAC1HDAC8
SCHEMBL16129641 0.85 MEN1 (0.66) ABCC1ABCB1MEN1KMT2AHDAC1
SCHEMBL18007313 0.84 PTPN1 (0.63) ABCC1MEN1KMT2AHDAC1HDAC8
SCHEMBL5724139 0.83 NAMPT (0.66) ABCC1MEN1KMT2ANAMPTALDH1A1
SCHEMBL16098533 0.81 ALDH1A1 (0.86) ABCB1MEN1KMT2ACYP3A4POLB
SCHEMBL18007302 0.80 MEN1 (0.65) ABCC1MEN1KMT2AHDAC8POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001766-B1 COMPOUNDS FOR THE TREATMENT OF CCR5-MEDIATED DISEASES SMITHKLINE BEECHAM CORP (US) 2003-04-09 EP disclosed
US-6515027-B1 Ligands, agonists or antagonists, of the CC chemokine receptor CC-CKR5 SMITHKLINE BEECHAM CORP. 2003-02-04 US disclosed