SCHEMBL6928237

SCHEMBL6928237

COC(=O)Nc1ccc(N)cc1OCCN(C(C)C)C(C)C

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 16/20 0.43
HTR2C P28335 1/20 0.43
SLC2A1 P11166 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6928801 0.81 PKM (0.62) GAAMAPTSMN1; SMN2
SCHEMBL4198415 0.76 GAA (0.55) MCHR1HTR2CSLC2A1GAAMAPT
SCHEMBL6204180 0.76 GAA (0.47) MCHR1HTR2CGAAMAPT
SCHEMBL6926905 0.76 MCHR1 (0.77) MCHR1HTR2CSLC2A1
SCHEMBL2071884 0.75 GAA (0.59) GAAMAPTSMN1; SMN2HPGD
SCHEMBL6922538 0.74 ALDH1A1 (0.41) MCHR1GAAMAPTSMN1; SMN2
Hydrochloric Acid SCHEMBL6926164 0.74 GAA (0.42) MCHR1HTR2CGAAMAPT
SCHEMBL6927859 0.73 GAA (0.41) MCHR1HTR2CGAAMAPT
SCHEMBL6927647 0.73 CYP1A2 (0.59) MCHR1HTR2CGAAMAPTSMN1; SMN2
SCHEMBL6807342 0.72 MCHR1 (0.48) MCHR1HTR2CGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001766-B1 COMPOUNDS FOR THE TREATMENT OF CCR5-MEDIATED DISEASES SMITHKLINE BEECHAM CORP (US) 2003-04-09 EP disclosed
US-6515027-B1 Ligands, agonists or antagonists, of the CC chemokine receptor CC-CKR5 SMITHKLINE BEECHAM CORP. 2003-02-04 US disclosed
EP-1001766-A4 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORP (US) 2001-04-04 EP disclosed
EP-1001766-A1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2000-05-24 EP disclosed
WO-1999001127-A1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 1999-01-14 WO disclosed