SCHEMBL6929093

SCHEMBL6929093

Cc1ccc(Cn2cncc2CO)cc1

nearest known ligand 0.66

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 18/20 0.66
CYP11B2 P19099 18/20 0.66
CYP19A1 P11511 2/20 0.45
TP53 P04637 1/20 0.43
MAPT P10636 1/20 0.43
LMNA P02545 1/20 0.43
HTT P42858 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
IDO1 P14902 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6599640 0.85 CYP11B1 (0.72) CYP11B1CYP11B2CYP19A1HTTSMN1; SMN2
SCHEMBL3820773 0.84 CYP11B1 (0.76) CYP11B1CYP11B2CYP19A1LMNAHTT
SCHEMBL6599385 0.84 CYP11B1 (0.48) CYP11B1CYP11B2CYP19A1
SCHEMBL6599480 0.83 CYP11B1 (0.73) CYP11B1CYP11B2CYP19A1IDO1
Hydrochloric Acid SCHEMBL6927027 0.83 CYP11B1 (0.49) CYP11B1CYP11B2CYP19A1TP53MAPT
SCHEMBL3079356 0.83 CYP11B1 (0.71) CYP11B1CYP11B2HTTIDO1
SCHEMBL6929673 0.83 CYP11B1 (0.75) CYP11B1CYP11B2IDO1
SCHEMBL3822319 0.82 CYP11B1 (0.52) CYP11B1CYP11B2CYP19A1TP53MAPT
SCHEMBL6926694 0.81 CYP11B1 (0.52) CYP11B1CYP11B2TP53MAPTLMNA
SCHEMBL3630524 0.80 CYP11B1 (1.00) CYP11B1CYP11B2CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1188407-C Imidazole derivatives with inhabiting activity to transterasa and preparing method thereof LG CHEMICAL LTD (KR) 2005-02-09 CN disclosed
EP-1045846-B1 IMIDAZOLE DERIVATIVES HAVING AN INHIBITORY ACTIVITY FOR FARNESYL TRANSFERASE AND PROCESS FOR PREPARATION THEREOF LG CHEMICAL LTD (KR) 2003-05-02 EP disclosed
US-6518429-B2 Anticancer agents, treating restenosis, atherosclerosis and hepatitis virus LG CHEMICAL, LTD. (KR) 2003-02-11 US disclosed
US-6472526-B1 SHOWS AN INHIBITORY ACTIVITY AGAINST FARNESYL TRANSFERASE OR PHARMACEUTICALLY ACCEPTABLE SALTS OR ISOMERS THEREOF, IN PHARMACEUTICAL COMPOSITION AND INTERMEDIATES LG CHEMICAL LTD. (KR) 2002-10-29 US disclosed
US-20020137769-A1 Imidazole derivatives having an inhibitory activity for farnesyl transferase and process for preparation thereof LG CHEMICAL LTD. 2002-09-26 US disclosed
US-6268363-B1 ANTITUMOR LG CHEMICAL LTD. (KR) 2001-07-31 US disclosed
CN-1279680-A Imidazole derivatives having farnesyl transferase inhibitory activity and process for producing the same LG CHEMICAL LTD (KR) 2001-01-10 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020137769-A1 Imidazole derivatives having an inhibitory activity for farnesyl transferase and process for preparation thereof FNTA, FNTB, FDPS CYP11B1 74/4885CYP11B2 110/4885CYP19A1 698/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.