SCHEMBL6929673

SCHEMBL6929673

COc1ccc(Cn2cncc2CO)cc1

nearest known ligand 0.75

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 15/20 0.75
CYP11B2 P19099 15/20 0.75
HSP90AA1 P07900 1/20 0.51
HSP90AB1 P08238 1/20 0.51
IDO1 P14902 1/20 0.46
GABRA5 P31644 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6599140 0.85 CYP11B1 (0.60) CYP11B1CYP11B2HSP90AA1HSP90AB1
Hydrochloric Acid SCHEMBL6924858 0.85 CYP11B1 (0.67) CYP11B1CYP11B2HSP90AA1HSP90AB1IDO1
SCHEMBL6929093 0.83 CYP11B1 (0.66) CYP11B1CYP11B2IDO1
SCHEMBL6599640 0.81 CYP11B1 (0.72) CYP11B1CYP11B2
SCHEMBL3873541 0.80 CYP11B2 (0.56) CYP11B1CYP11B2
SCHEMBL6599480 0.80 CYP11B1 (0.73) CYP11B1CYP11B2IDO1
SCHEMBL3079356 0.79 CYP11B1 (0.71) CYP11B1CYP11B2HSP90AA1HSP90AB1IDO1
SCHEMBL15507125 0.78 CYP11B1 (0.61) CYP11B1CYP11B2HSP90AA1HSP90AB1IDO1
SCHEMBL7981213 0.78 CYP11B1 (0.73) CYP11B1CYP11B2
SCHEMBL28941444 0.78 CYP11B1 (0.61) CYP11B1CYP11B2HSP90AA1HSP90AB1IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1188407-C Imidazole derivatives with inhabiting activity to transterasa and preparing method thereof LG CHEMICAL LTD (KR) 2005-02-09 CN disclosed
EP-1045846-B1 IMIDAZOLE DERIVATIVES HAVING AN INHIBITORY ACTIVITY FOR FARNESYL TRANSFERASE AND PROCESS FOR PREPARATION THEREOF LG CHEMICAL LTD (KR) 2003-05-02 EP disclosed
US-6518429-B2 Anticancer agents, treating restenosis, atherosclerosis and hepatitis virus LG CHEMICAL, LTD. (KR) 2003-02-11 US disclosed
US-6472526-B1 SHOWS AN INHIBITORY ACTIVITY AGAINST FARNESYL TRANSFERASE OR PHARMACEUTICALLY ACCEPTABLE SALTS OR ISOMERS THEREOF, IN PHARMACEUTICAL COMPOSITION AND INTERMEDIATES LG CHEMICAL LTD. (KR) 2002-10-29 US disclosed
US-20020137769-A1 Imidazole derivatives having an inhibitory activity for farnesyl transferase and process for preparation thereof LG CHEMICAL LTD. 2002-09-26 US disclosed
US-6268363-B1 ANTITUMOR LG CHEMICAL LTD. (KR) 2001-07-31 US disclosed
CN-1279680-A Imidazole derivatives having farnesyl transferase inhibitory activity and process for producing the same LG CHEMICAL LTD (KR) 2001-01-10 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020137769-A1 Imidazole derivatives having an inhibitory activity for farnesyl transferase and process for preparation thereof FNTA, FNTB, FDPS CYP11B1 74/4885CYP11B2 110/4885HSP90AA1 2008/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.