SCHEMBL6929762

SCHEMBL6929762

CC(C)OCCOS(=O)(=O)c1ccc(Br)cc1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.43
LMNA P02545 1/20 0.40
PLCG1 P19174 1/20 0.40
CA2 P00918 3/20 0.37
GAA P10253 2/20 0.37
TSHR P16473 1/20 0.36
MMP2 P08253 3/20 0.35
MMP1 P03956 2/20 0.35
MMP9 P14780 2/20 0.35
MMP13 P45452 2/20 0.35
MMP3 P08254 1/20 0.35
MMP7 P09237 1/20 0.35
POLB P06746 1/20 0.35
CA12 O43570 1/20 0.34
CA9 Q16790 1/20 0.34
CA1 P00915 1/20 0.34
MMP8 P22894 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11222461 0.86 PLCG1 (0.52) ALDH1A1LMNAPLCG1CA2GAA
SCHEMBL57438 0.85 CA12 (0.45) ALDH1A1LMNACA2GAATSHR
SCHEMBL9182366 0.81 PLCG1 (0.44) ALDH1A1LMNAPLCG1CA2GAA
SCHEMBL27649868 0.79 PLCG1 (0.45) PLCG1CA2GAATSHRMMP2
SCHEMBL19523745 0.78 GAA (0.44) PLCG1CA2GAAMMP2MMP1
SCHEMBL6601720 0.78 GAA (0.44) LMNAPLCG1CA2GAATSHR
SCHEMBL3386673 0.77 PLCG1 (0.48) PLCG1CA2GAAMMP2MMP1
SCHEMBL19229836 0.76 CA2 (0.46) ALDH1A1PLCG1CA2GAATSHR
SCHEMBL2564478 0.75 CYP3A4 (0.46) ALDH1A1GAATSHRCA12CA9
SCHEMBL10433465 0.75 PLCG1 (0.39) ALDH1A1PLCG1CA2GAAMMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6518282-B1 Treatment of pruritic dermatoses including allergic dermatitis and atopy in animals and humans PFIZER INC. 2003-02-11 US disclosed
EP-1072595-A2 4-arylpiperidine derivatives for the treatment of pruritus PFIZER INC. (US) 2001-01-31 EP disclosed