SCHEMBL693144

SCHEMBL693144

CCOc1cccc([C@H](CC(=O)O)NC(=O)Nc2c(O)c(C)cn(Cc3c(C)cccc3Cl)c2=O)c1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.37
ALDH1A1 P00352 3/20 0.37
FFAR1 O14842 3/20 0.37
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
PYGL P06737 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
SLC22A12 Q96S37 1/20 0.34
CTSA P10619 3/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
ITGB1 P05556 2/20 0.33
ITGA4 P13612 2/20 0.33
HPGD P15428 1/20 0.33
LCK P06239 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL686989 0.94 SMN1; SMN2 (0.38) KDM4EALDH1A1FFAR1CYP2C9CYP2C19
SCHEMBL688501 0.93 SMN1; SMN2 (0.40) KDM4EALDH1A1FFAR1CYP3A4CYP2C9
SCHEMBL686996 0.92 P2RX3 (0.35) KDM4EALDH1A1FFAR1CYP3A4CYP2C9
SCHEMBL687688 0.91 SMN1; SMN2 (0.37) KDM4EALDH1A1FFAR1CYP3A4CYP2C9
SCHEMBL688167 0.91 SMN1; SMN2 (0.43) KDM4EALDH1A1CYP3A4CYP2C9CYP2C19
SCHEMBL687744 0.91 PTGER3 (0.43) FFAR1NPSR1RXFP1SLC22A12CTSA
SCHEMBL688946 0.91 SMN1; SMN2 (0.34) KDM4EALDH1A1FFAR1CYP2C9CYP2C19
SCHEMBL688507 0.90 SMN1; SMN2 (0.38) KDM4EALDH1A1FFAR1CYP3A4CYP2C9
SCHEMBL687802 0.89 CTSA (0.34) KDM4EALDH1A1FFAR1CYP3A4CYP2C9
SCHEMBL687119 0.89 SMN1; SMN2 (0.36) KDM4EALDH1A1FFAR1CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203766-B1 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS INC (US) 2012-02-29 EP disclosed
EP-1203766-A2 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors TEXAS BIOTECHNOLOGY CORPORATION (US) 2002-05-08 EP disclosed