SCHEMBL6933270

SCHEMBL6933270

C/C(O)=C(\C#N)CC(=O)O

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LDHA P00338 1/20 0.38
SRR Q9GZT4 1/20 0.38
DHODH Q02127 2/20 0.32
KDM4E B2RXH2 2/20 0.31
KDM5C P41229 2/20 0.31
EGLN1 Q9GZT9 2/20 0.31
PHF8 Q9UPP1 2/20 0.31
KDM2A Q9Y2K7 2/20 0.31
MCL1 Q07820 1/20 0.31
KDM6B O15054 1/20 0.31
LMNA P02545 1/20 0.31
SLC15A2 Q16348 1/20 0.31
FFAR3 O14843 1/20 0.30
CTH P32929 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6933272 1.00 LDHA (0.38) LDHASRRDHODHKDM4EKDM5C
Trifluoroacetic Acid SCHEMBL27543172 0.88 DHODH (0.36) DHODH
SCHEMBL11456377 0.75 ALDH1A1 (0.38) LDHASRRLMNA
SCHEMBL8940378 0.74
Acetoacetic Acid SCHEMBL28196823 0.69 KDM4E (0.44) LDHASRRKDM4EKDM5CEGLN1
SCHEMBL7880615 0.67
SCHEMBL11013811 0.67 LDHA (0.40) LDHASRRKDM4EKDM5CEGLN1
Acetoacetic Acid SCHEMBL14332619 0.66
Acetoacetic Acid SCHEMBL10916658 0.66
Acetic Acid SCHEMBL3939078 0.65 FFAR3 (0.41) LDHASRRMCL1FFAR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0859000-B1 Isoxazole amide and crotonamid derivatives and drug and diagnostic uses thereof AVENTIS PHARMA GMBH (DE) 2003-01-22 EP claimed
US-5977151-A ANTITUMOR HOECHST AKTIENGESELLSCHAFT (DE) 1999-11-02 US claimed
US-6265588-B1 USE AS PHARMACEUTICALS; AS AN ANTIGEN FOR PRODUCTION OF ANTIBODIES AND IN DIAGNOSIS AND PURIFICATION AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2001-07-24 US disclosed
US-6121479-A ANTIINFLAMMATORY AND ANTICARCINOGENIC AGENTS; AUTOIMMUNE DISEASES HOECHST AKTIENGESELLSCHAFT (DE) 2000-09-19 US disclosed
US-5977151-A ANTITUMOR HOECHST AKTIENGESELLSCHAFT (DE) 1999-11-02 US disclosed