SCHEMBL6934308

SCHEMBL6934308

COc1ccc([C@@H](N)CC(=O)OC(C)(C)C)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C19 P33261 1/20 0.49
NPSR1 Q6W5P4 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.42
MMP1 P03956 1/20 0.41
FFAR1 O14842 1/20 0.40
AOC3 Q16853 2/20 0.40
OPRD1 P41143 1/20 0.39
TNF P01375 1/20 0.39
GRM8 O00222 1/20 0.39
GRM6 O15303 1/20 0.39
GRM4 Q14833 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
LMNA P02545 1/20 0.39
KDM4E B2RXH2 2/20 0.39
MAPT P10636 1/20 0.39
ESR2 Q92731 1/20 0.39
ALDH1A1 P00352 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14698374 0.84 MIF (0.37) CYP1A2CYP2D6CYP2C19LMNAMAPT
SCHEMBL14698215 0.84 MIF (0.37) CYP1A2CYP2D6CYP2C19LMNAMAPT
SCHEMBL5720903 0.84 ACHE (0.39) CYP2D6CYP2C19L3MBTL1FFAR1OPRD1
SCHEMBL2294181 0.84 CYP1A2 (0.54) CYP1A2CYP2D6CYP2C19NPSR1L3MBTL1
SCHEMBL469053 0.83 CTSS (0.42) L3MBTL1CA2MAPTALDH1A1HSD17B10
Hydrochloric Acid SCHEMBL8323812 0.83 CYP1A2 (0.53) CYP1A2CYP2D6CYP2C19NPSR1L3MBTL1
SCHEMBL1573827 0.83 CTSS (0.42) L3MBTL1CA2MAPTALDH1A1HSD17B10
SCHEMBL1952090 0.83 CTSS (0.42) L3MBTL1CA2MAPTALDH1A1HSD17B10
Hydrochloric Acid SCHEMBL6692761 0.83 CYP1A2 (0.53) CYP1A2CYP2D6CYP2C19NPSR1L3MBTL1
SCHEMBL28393121 0.82 DPP4 (0.50) CYP2C19CA1CA2MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0918059-B1 Substituted imidazoline derivatives, their preparation, their use, and pharmaceutical compositions containing them AVENTIS PHARMA GMBH (DE) 2003-06-25 EP disclosed
EP-0918059-A1 Substituted imidazoline derivatives, their preparation, their use, and pharmaceutical compositions containing them Hoechst Marion Roussel Deutschland GmbH (DE) 1999-05-26 EP disclosed