SCHEMBL6935740

SCHEMBL6935740

COC(=NN[C@@H](CC(=O)O)C(N)=O)NC(=O)c1cccc(NC(=N)N)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 5/20 0.46
ITGA2B P08514 2/20 0.46
PARP1 P09874 1/20 0.45
PARP10 Q53GL7 1/20 0.45
ITGAV P06756 3/20 0.40
PLK4 O00444 1/20 0.40
CHEK1 O14757 1/20 0.40
AURKA O14965 1/20 0.40
CHUK O15111 1/20 0.40
DAPK3 O43293 1/20 0.40
JAK2 O60674 1/20 0.40
ROCK2 O75116 1/20 0.40
PAK4 O96013 1/20 0.40
CHEK2 O96017 1/20 0.40
CDK1 P06493 1/20 0.40
PIM1 P11309 1/20 0.40
PRKACA P17612 1/20 0.40
FGFR3 P22607 1/20 0.40
RPS6KB1 P23443 1/20 0.40
CDK2 P24941 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6938674 0.85 KMT2A (0.39) ITGB3ITGA2BPARP1PARP10ALDH1A1
SCHEMBL6934969 0.79 ITGB3 (0.51) ITGB3ITGA2BPARP1PARP10ITGAV
SCHEMBL30083944 0.75 ITGB3 (0.51) ITGB3ITGA2BPARP1PARP10ITGAV
SCHEMBL7879691 0.75 ITGB3 (0.56) ITGB3ITGA2BPARP1PARP10ITGAV
SCHEMBL18271386 0.73 ITGB3 (0.49) ITGB3ITGA2BPARP1PARP10ITGAV
SCHEMBL7315631 0.72 ITGB3 (0.50) ITGB3ITGA2BPARP1PARP10ITGAV
SCHEMBL6938684 0.70 ITGB3 (0.43) ITGB3ITGA2BPARP1PARP10ITGAV
SCHEMBL18269210 0.70 ITGB3 (0.48) ITGB3ITGA2BPARP1PARP10ITGAV
SCHEMBL7452316 0.70 ITGB3 (0.57) ITGB3ITGA2BPARP1PARP10PLK4
SCHEMBL9335947 0.70 ITGB3 (0.69) ITGB3ITGA2BPARP1ITGAVPLAU

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6326403-B1 CARDIOVASCULAR DISORDERS MERCK PATENT GESELLSCHAFT MIT (DE) 2001-12-04 US claimed
EP-1097127-B1 DIACYLHYDRAZINE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GMBH (DE) 2003-03-12 EP disclosed
US-6326403-B1 CARDIOVASCULAR DISORDERS MERCK PATENT GESELLSCHAFT MIT (DE) 2001-12-04 US disclosed