SCHEMBL6936458

SCHEMBL6936458

NC(=O)c1cn(C[C@H](CCCn2c(=O)sc3ccccc32)OCc2ccccc2)cn1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 5/20 0.43
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
CYP3A4 P08684 3/20 0.43
CYP2D6 P10635 3/20 0.43
CYP2C19 P33261 3/20 0.43
CYP1A2 P05177 2/20 0.43
CYP2C9 P11712 2/20 0.43
HTT P42858 2/20 0.41
TSHR P16473 2/20 0.41
HTR1A P08908 1/20 0.40
HTR7 P34969 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
ALDH1A1 P00352 1/20 0.39
MAPK1 P28482 1/20 0.39
ATM Q13315 1/20 0.39
HPGD P15428 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
KDM4E B2RXH2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6942807 0.84 L3MBTL1 (0.44) L3MBTL1NPC1RAB9ASMN1; SMN2CYP3A4
SCHEMBL5671897 0.81 ADA (0.47) CYP2D6CYP2C19CYP1A2CYP2C9
SCHEMBL6169457 0.81 ADA (0.49)
SCHEMBL6939156 0.80 ADA (0.46)
SCHEMBL6169467 0.80 ADA (0.48)
SCHEMBL6935843 0.79 KMO (0.40) NPC1RAB9ASMN1; SMN2
SCHEMBL7072052 0.78 MAPT (0.45) L3MBTL1SMN1; SMN2HTTTSHRALDH1A1
SCHEMBL6936452 0.78 ADA (0.42) L3MBTL1NPC1RAB9ASMN1; SMN2CYP3A4
SCHEMBL6171160 0.75 ADA (0.44)
SCHEMBL6171261 0.75 ADA (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6596738-B1 Inhibiting activity to adenosine deaminase (hereinafter described as ADA) An adenosine deaminase inhibiting agent comprising a compound of the formula (I): FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-07-22 US disclosed