SCHEMBL6937376

SCHEMBL6937376

O=C(O)Oc1ccc(NC(=O)OCC2c3ccccc3-c3ccccc32)nc1

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.49
KMT2A Q03164 2/20 0.46
FABP5 Q01469 3/20 0.40
FABP7 O15540 2/20 0.40
MDM4 O15151 1/20 0.40
TP53 P04637 1/20 0.40
CASP3 P42574 2/20 0.40
MDM2 Q00987 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7872045 0.84 HCAR3 (0.51) EPHX2KMT2AFABP5FABP7MDM4
SCHEMBL28552605 0.82 EPHX2 (0.52) EPHX2KMT2ATP53MDM2
SCHEMBL21303577 0.79 EPHX2 (0.56) EPHX2KMT2AFABP5FABP7
SCHEMBL8366872 0.75 EPHX2 (0.75) EPHX2KMT2AFABP5FABP7CASP3
SCHEMBL27644637 0.74 EPHX2 (0.59) EPHX2KMT2ACASP3
SCHEMBL15387199 0.74 MDM2 (0.47) EPHX2KMT2AMDM4TP53CASP3
SCHEMBL346077 0.73 KMT2A (0.52) EPHX2KMT2AFABP5FABP7MDM4
SCHEMBL31370380 0.72 MDM4 (0.49) MDM4TP53CASP3MDM2
SCHEMBL25253846 0.72 MDM2 (0.52) MDM4TP53CASP3MDM2
SCHEMBL13688459 0.72 KMT2A (0.62) EPHX2KMT2AFABP5FABP7MDM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1097127-B1 DIACYLHYDRAZINE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GMBH (DE) 2003-03-12 EP disclosed
EP-1097127-A1 DIACYLHYDRAZINE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GmbH (DE) 2001-05-09 EP disclosed
WO-2000003973-A1 DIACYLHYDRAZINE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GMBH (DE) 2000-01-27 WO disclosed