SCHEMBL6940969

SCHEMBL6940969

CCC(c1cc(N)ccc1N)c1cc(N)ccc1N

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 3/20 0.38
MAPT P10636 6/20 0.36
MEN1 O00255 6/20 0.36
KMT2A Q03164 6/20 0.36
TDP1 Q9NUW8 4/20 0.36
POLB P06746 3/20 0.36
USP2 O75604 3/20 0.36
THRB P10828 3/20 0.36
PKM P14618 2/20 0.36
BLM P54132 2/20 0.36
RECQL P46063 2/20 0.36
APEX1 P27695 1/20 0.36
MCL1 Q07820 1/20 0.36
ALDH1A1 P00352 8/20 0.36
GAA P10253 6/20 0.36
KDM4E B2RXH2 4/20 0.36
TP53 P04637 2/20 0.36
HTT P42858 2/20 0.36
CASP7 P55210 1/20 0.36
ATM Q13315 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL111964 0.83 CASP1 (0.43) CASP1MAPTMEN1KMT2ATDP1
SCHEMBL3187941 0.83 CASP1 (0.38) CASP1MAPTMEN1KMT2ATDP1
Hydrochloric Acid SCHEMBL8334339 0.81 GAA (0.39) CASP1MAPTMEN1KMT2ATDP1
SCHEMBL249358 0.81 ALDH1A1 (0.43) CASP1MAPTMEN1KMT2ATDP1
SCHEMBL30120579 0.79 PDE2A (0.39) CASP1MAPTMEN1KMT2ATDP1
SCHEMBL11402718 0.79 PDE2A (0.39) CASP1MAPTMEN1KMT2ATDP1
SCHEMBL28258130 0.77 ALDH1A1 (0.48) CASP1MAPTMEN1KMT2ATDP1
SCHEMBL6920084 0.76 CASP1 (0.33) CASP1MAPTMEN1KMT2ATDP1
Benzene SCHEMBL27545048 0.76 ANPEP (0.41) CASP1MAPTMEN1KMT2ATDP1
SCHEMBL1299720 0.75 CYP3A4 (0.47) CASP1MAPTTDP1POLBTHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1301163-A1 OXIDISED HAIR COLOURING AGENTS CONTAINING AT LEAST ONE DISUBSTITUITED 2.4-DIAMINO PHENYL ETHER AS A COUPLING COMPONENT Henkel Kommanditgesellschaft auf Aktien (DE) 2003-04-16 EP claimed
WO-2002005767-A1 OXIDISED HAIR COLOURING AGENTS CONTAINING AT LEAST ONE DISUBSTITUITED 2.4-DIAMINO PHENYL ETHER AS A COUPLING COMPONENT HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2002-01-24 WO claimed
EP-1301163-A1 OXIDISED HAIR COLOURING AGENTS CONTAINING AT LEAST ONE DISUBSTITUITED 2.4-DIAMINO PHENYL ETHER AS A COUPLING COMPONENT Henkel Kommanditgesellschaft auf Aktien (DE) 2003-04-16 EP disclosed
WO-2002005767-A1 OXIDISED HAIR COLOURING AGENTS CONTAINING AT LEAST ONE DISUBSTITUITED 2.4-DIAMINO PHENYL ETHER AS A COUPLING COMPONENT HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2002-01-24 WO disclosed