SCHEMBL6942540

SCHEMBL6942540

N#Cc1ccc([N+](=O)[O-])cc1-c1ccccc1N.N#Cc1ccc([N+](=O)[O-])cc1Cl

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VCAM1 P19320 2/20 0.52
PDE7A Q13946 3/20 0.48
HSD17B10 Q99714 1/20 0.42
RORC P51449 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
POLB P06746 1/20 0.41
PTPRC P08575 2/20 0.40
BCHE P06276 1/20 0.40
ACHE P22303 1/20 0.40
CES1 P23141 1/20 0.40
S100A4 P26447 1/20 0.40
CASP3 P42574 1/20 0.40
SENP8 Q96LD8 1/20 0.40
SENP7 Q9BQF6 1/20 0.40
SENP6 Q9GZR1 1/20 0.40
NPBWR1 P48145 1/20 0.39
KMT2A Q03164 2/20 0.39
ALDH1A1 P00352 3/20 0.39
MEN1 O00255 1/20 0.39
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5900973 0.92 VCAM1 (0.49) VCAM1PDE7ASMN1; SMN2POLBPTPRC
SCHEMBL2477528 0.82 VCAM1 (0.74) VCAM1PDE7AHSD17B10SMN1; SMN2KMT2A
SCHEMBL7571256 0.74 VCAM1 (0.47) VCAM1SMN1; SMN2POLBPTPRCBCHE
SCHEMBL1706658 0.73 VCAM1 (0.59) VCAM1SMN1; SMN2KMT2AALDH1A1MEN1
Dinitrophenylene SCHEMBL27564017 0.72 VCAM1 (0.68) VCAM1HSD17B10SMN1; SMN2ACHECES1
Dinitrophenylene SCHEMBL27864502 0.72 TSHR (0.57) VCAM1SMN1; SMN2ACHECES1CASP3
SCHEMBL689735 0.71 VCAM1 (0.66) VCAM1SMN1; SMN2CASP3SENP8SENP7
SCHEMBL2649876 0.70 VCAM1 (0.49) VCAM1SMN1; SMN2PTPRCBCHEACHE
Nitrogen SCHEMBL28796067 0.70 VCAM1 (0.64) VCAM1SMN1; SMN2CASP3SENP8SENP7
SCHEMBL892830 0.70 VCAM1 (1.00) VCAM1HSD17B10SMN1; SMN2KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1233950-A4 3,4-DIHYDRO-(1H)QUINAZOLIN-2-ONE COMPOUNDS AS CSBP/P39 kINASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2003-03-26 EP disclosed
EP-1233950-A1 3,4-DIHYDRO-(1H)QUINAZOLIN-2-ONE COMPOUNDS AS CSBP/P39 kINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2002-08-28 EP disclosed
WO-2001038313-A1 3,4-DIHYDRO-(1H)QUINAZOLIN-2-ONE COMPOUNDS AS CSBP/p39 kINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (GB) 2001-05-31 WO disclosed