SCHEMBL6942601

SCHEMBL6942601

CC(C)(C)[Si](C)(C)OC[C@@H](O)CCn1ccc2ccc([N+](=O)[O-])cc21

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 1/20 0.45
AR P10275 1/20 0.38
ADRB2 P07550 4/20 0.36
ADRB1 P08588 4/20 0.36
ADRB3 P13945 4/20 0.36
CDC7 O00311 1/20 0.35
MTNR1A P48039 2/20 0.33
MTNR1B P49286 2/20 0.33
MAPT P10636 1/20 0.33
ADA P00813 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6942605 1.00 HTR7 (0.45) HTR7ARADRB2ADRB1ADRB3
SCHEMBL4511606 0.84 HTR7 (0.51) HTR7ARCDC7MTNR1AMTNR1B
SCHEMBL6940163 0.82 ADRB2 (0.41) ADRB2ADRB1ADRB3MAPT
SCHEMBL6940159 0.82 ADRB2 (0.41) ADRB2ADRB1ADRB3MAPT
SCHEMBL6933495 0.80 ADA (0.56) HTR7ADA
SCHEMBL6933500 0.80 CDK4 (0.45) MAPT
SCHEMBL6933502 0.80 CDK4 (0.45) MAPT
SCHEMBL6938432 0.76 HTR7 (0.49) HTR7MAPTADA
SCHEMBL6938431 0.76 HTR7 (0.49) HTR7MAPTADA
Ammonia Solution, Strong SCHEMBL27732810 0.74 HTR7 (0.57) HTR7ARCDC7MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6596738-B1 Inhibiting activity to adenosine deaminase (hereinafter described as ADA) An adenosine deaminase inhibiting agent comprising a compound of the formula (I): FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-07-22 US disclosed
EP-1161429-A2 HETEROCYCLIC COMPOUNDS AS ADENOSINE DEAMINASE INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-12-12 EP disclosed
WO-2000055155-A2 HETEROCYCLIC COMPOUNDS AS ADENOSINE DEAMINASE INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-09-21 WO disclosed