SCHEMBL6943341

SCHEMBL6943341

O=C(O)C(=O)CC(=O)c1cc(Cc2ccccc2)ccc1OC(F)C(F)F

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ERCC5 P28715 7/20 0.42
FEN1 P39748 7/20 0.42
PTPN1 P18031 5/20 0.42
HAO1 Q9UJM8 1/20 0.41
HNF4A P41235 1/20 0.41
MPO P05164 1/20 0.38
PDE4A P27815 2/20 0.37
PDE4B Q07343 2/20 0.37
PDE4C Q08493 2/20 0.37
PDE4D Q08499 2/20 0.37
CFD P00746 1/20 0.36
PPARG P37231 3/20 0.36
PPARA Q07869 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5148099 0.85 IDO1 (0.44) ERCC5FEN1PTPN1HAO1HNF4A
Dimethylamine SCHEMBL6950061 0.84 IDO1 (0.44) ERCC5FEN1PTPN1HAO1HNF4A
SCHEMBL6948223 0.81 NPC1 (0.47) ERCC5FEN1PTPN1HAO1HNF4A
SCHEMBL6948028 0.80 HAO1 (0.39) ERCC5FEN1PTPN1HAO1HNF4A
SCHEMBL6945630 0.80 HAO1 (0.42) ERCC5FEN1PTPN1HAO1HNF4A
SCHEMBL6943337 0.80 ALDH1A1 (0.46) ERCC5FEN1PTPN1HAO1HNF4A
SCHEMBL6946203 0.79 LMNA (0.46) ERCC5FEN1PTPN1HAO1HNF4A
SCHEMBL6950546 0.79 PDE4A (0.42) ERCC5FEN1PTPN1HAO1HNF4A
SCHEMBL6951239 0.78 HAO1 (0.43) ERCC5FEN1PTPN1HAO1HNF4A
Dimethylamine SCHEMBL6947623 0.78 LMNA (0.46) ERCC5FEN1PTPN1HAO1HNF4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US claimed
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP disclosed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US disclosed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP disclosed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO disclosed