SCHEMBL6943570

SCHEMBL6943570

CN(C)c1cc(Cc2ccccc2Cl)cc(C(=O)CC(=O)C(=O)O)c1

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 3/20 0.48
KDM4E B2RXH2 1/20 0.47
LMNA P02545 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
FEN1 P39748 12/20 0.44
ERCC5 P28715 11/20 0.44
HAO1 Q9UJM8 2/20 0.43
MRGPRX4 Q96LA9 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6946034 0.85 PTPN1 (0.53) PTPN1FEN1ERCC5HAO1
SCHEMBL6951641 0.81 FEN1 (0.54) PTPN1LMNASMN1; SMN2FEN1ERCC5
Dimethylamine SCHEMBL6943573 0.81 PTPN1 (0.69) PTPN1FEN1ERCC5HAO1
SCHEMBL6947650 0.80 PTPN1 (0.72) PTPN1FEN1ERCC5HAO1
SCHEMBL6943298 0.77 PTPN1 (0.46) PTPN1KDM4EFEN1ERCC5HAO1
SCHEMBL6949821 0.72 PTPN1 (0.64) PTPN1LMNAFEN1ERCC5HAO1
SCHEMBL6946193 0.72 PTPN1 (0.67) PTPN1SMN1; SMN2FEN1ERCC5HAO1
SCHEMBL6947604 0.71 ERCC5 (0.61) PTPN1LMNAFEN1ERCC5HAO1
SCHEMBL6947985 0.70 PTPN1 (0.64) PTPN1FEN1ERCC5HAO1
SCHEMBL6946220 0.70 PTPN1 (0.71) PTPN1FEN1ERCC5HAO1MRGPRX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP claimed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US claimed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP claimed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO claimed
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP disclosed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US disclosed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP disclosed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO disclosed