SCHEMBL6943787

SCHEMBL6943787

O=C(O)/C(O)=C/C(=O)c1cccc(N(Cc2ccccc2)Cc2ccccc2)c1

nearest known ligand 0.61

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 4/20 0.61
CRHBP P24387 1/20 0.52
CRHR2 Q13324 1/20 0.52
ALDH1A1 P00352 1/20 0.47
LMNA P02545 1/20 0.47
KMT2A Q03164 4/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
NR3C1 P04150 1/20 0.43
MEN1 O00255 3/20 0.42
GRM2 Q14416 1/20 0.40
SLC16A3 O15427 1/20 0.40
SLC16A1 P53985 1/20 0.40
MTNR1A P48039 1/20 0.39
MTNR1B P49286 1/20 0.39
TMEM97 Q5BJF2 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
GPR52 Q9Y2T5 1/20 0.39
TDP1 Q9NUW8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6943789 1.00 PTPN1 (0.61) PTPN1CRHBPCRHR2ALDH1A1LMNA
SCHEMBL6943582 0.84 CYP2C19 (0.47) PTPN1CRHBPCRHR2KMT2ANR3C1
SCHEMBL6943247 0.84 CYP2C19 (0.47) PTPN1CRHBPCRHR2KMT2ANR3C1
SCHEMBL6952400 0.81 PTPN1 (0.68) PTPN1CRHBPCRHR2ALDH1A1LMNA
SCHEMBL1375356 0.78 PRSS1 (0.50) PTPN1ALDH1A1LMNAGPR52TDP1
SCHEMBL28458480 0.78 PTPN1 (0.65) PTPN1CRHBPCRHR2ALDH1A1LMNA
SCHEMBL22658227 0.78 CRHBP (0.68) PTPN1CRHBPCRHR2ALDH1A1LMNA
SCHEMBL1375355 0.78 PRSS1 (0.50) PTPN1ALDH1A1LMNAGPR52TDP1
SCHEMBL4598475 0.78 CRHBP (0.59) PTPN1CRHBPCRHR2ALDH1A1LMNA
SCHEMBL4598473 0.78 CRHBP (0.59) PTPN1CRHBPCRHR2ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP claimed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US claimed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP claimed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO claimed
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP disclosed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US disclosed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP disclosed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO disclosed