SCHEMBL6943886

SCHEMBL6943886

C=CCOC(=O)[C@H](CC(C)C)[C@H](OCc1ccccc1)C(=O)OC

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 6/20 0.41
PSMB5 P28074 1/20 0.40
CTSK P43235 4/20 0.40
CTSB P07858 1/20 0.39
SLC1A3 P43003 2/20 0.39
SLC1A2 P43004 2/20 0.39
SLC1A1 P43005 2/20 0.39
MEN1 O00255 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
KMT2A Q03164 1/20 0.39
MMP2 P08253 6/20 0.39
MMP3 P08254 6/20 0.39
MMP7 P09237 5/20 0.39
MMP8 P22894 2/20 0.39
ADAM17 P78536 1/20 0.39
CTSL P07711 1/20 0.39
MMP9 P14780 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6943883 1.00 MMP1 (0.41) MMP1PSMB5CTSKCTSBSLC1A3
SCHEMBL6946515 0.84 SLC1A3 (0.49) MMP1PSMB5CTSKCTSBSLC1A3
SCHEMBL6946518 0.84 SLC1A3 (0.49) MMP1PSMB5CTSKCTSBSLC1A3
SCHEMBL2000458 0.75 KMT2A (0.53) SLC1A3SLC1A2SLC1A1MEN1CYP1A2
SCHEMBL4011033 0.75 KMT2A (0.53) SLC1A3SLC1A2SLC1A1MEN1CYP1A2
SCHEMBL8622116 0.75 SLC1A3 (0.50) PSMB5CTSKCTSBSLC1A3SLC1A2
SCHEMBL8622114 0.75 SLC1A3 (0.50) PSMB5CTSKCTSBSLC1A3SLC1A2
SCHEMBL8496632 0.73 PSMB5 (0.55) PSMB5CTSKCTSBCTSL
SCHEMBL8679705 0.73 SLC1A2 (0.67) SLC1A3SLC1A2SLC1A1MEN1CYP1A2
SCHEMBL8678574 0.73 SLC1A2 (0.67) SLC1A3SLC1A2SLC1A1MEN1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0993442-B1 HYDRAZINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2003-04-23 EP disclosed
US-6235787-B1 ANTIINFLAMMATORY AGENTS; RHEUMATIC DISEASES; BONE DISORDERS; SKIN DISORDERS; MULTIPLE SCLEROSIS HOFFMANN-LA ROCHE INC. 2001-05-22 US disclosed
EP-0993442-A1 HYDRAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2000-04-19 EP disclosed
WO-1999001428-A1 HYDRAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1999-01-14 WO disclosed