SCHEMBL6944966

SCHEMBL6944966

COCC(=O)c1cc(Cc2ccccc2)cc(CN(C)C)c1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.42
TSHR P16473 1/20 0.42
LMNA P02545 2/20 0.40
MAPK1 P28482 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
CASP3 P42574 1/20 0.39
SENP7 Q9BQF6 1/20 0.39
SENP6 Q9GZR1 1/20 0.39
ACHE P22303 3/20 0.39
BCHE P06276 2/20 0.39
EGFR P00533 3/20 0.39
LTA4H P09960 4/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
MCHR1 Q99705 1/20 0.38
THRA P10827 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6951262 0.81 LTA4H (0.47) ALDH1A1LMNAMAPK1L3MBTL1CASP3
Dimethylamine SCHEMBL6944970 0.80 KDM4E (0.44) ALDH1A1LMNAMAPK1L3MBTL1CASP3
Benzene SCHEMBL28216395 0.70 KMT2A (0.56) ALDH1A1TSHRLMNAMAPK1L3MBTL1
SCHEMBL54072 0.70 KMT2A (0.56) ALDH1A1TSHRLMNAMAPK1L3MBTL1
Diphenylmethane SCHEMBL28227772 0.70 TSHR (0.85) ALDH1A1TSHRLMNALTA4HSMN1; SMN2
SCHEMBL9636764 0.69 TSHR (0.68) ALDH1A1TSHRLMNAMAPK1ACHE
SCHEMBL27916834 0.69 PLA2G10 (0.53) TSHRLMNAMEN1KMT2A
Hydrochloric Acid SCHEMBL27547476 0.69 NPC1 (0.54) ALDH1A1TSHRLMNAMAPK1L3MBTL1
SCHEMBL8399349 0.69 NPC1 (0.54) ALDH1A1TSHRLMNAMAPK1L3MBTL1
SCHEMBL6949247 0.68 LTA4H (0.43) ALDH1A1LMNAMAPK1L3MBTL1CASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP disclosed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US disclosed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP disclosed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO disclosed