SCHEMBL6945196

SCHEMBL6945196

Cc1nnn(Cc2ccc3[nH]cc(CCCCN(C)C)c3c2)n1

nearest known ligand 0.60

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 13/20 0.59
HTR2C P28335 10/20 0.59
HTR1D P28221 2/20 0.51
HTR1B P28222 2/20 0.51
ADRA2C P18825 1/20 0.51
HTR2A P28223 1/20 0.51
HRH1 P35367 1/20 0.51
HTR2B P41595 1/20 0.51
SLC6A4 P31645 5/20 0.49
MPO P05164 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6945655 0.79 HTR1A (0.60) HTR1AHTR2CHTR1DHTR1BADRA2C
SCHEMBL6939216 0.76 HTR1A (0.65) HTR1AHTR2CHTR1DHTR1BADRA2C
SCHEMBL8783747 0.74 HTR1A (1.00) HTR1AHTR2CHTR1DHTR1BADRA2C
SCHEMBL27392904 0.73 HTR1A (0.67) HTR1AHTR2CHTR1DHTR1BADRA2C
SCHEMBL6942548 0.72 HTR1A (0.52) HTR1AHTR2CHTR1DHTR1BADRA2C
SCHEMBL8784514 0.72 HTR1A (1.00) HTR1AHTR2CHTR1DHTR1BADRA2C
SCHEMBL6944315 0.71 SLC6A4 (0.49) HTR1AHTR2CHTR1DHTR1BADRA2C
SCHEMBL6941530 0.71 HTR1A (0.75) HTR1AHTR2CHTR1DHTR1BADRA2C
SCHEMBL6944313 0.70 HTR1A (0.55) HTR1AHTR2CHTR1DHTR1BSLC6A4
SCHEMBL8784534 0.70 HTR1A (1.00) HTR1AHTR2CHTR1DHTR1BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0925302-B1 PALLADIUM CATALYZED INDOLIZATION MERCK & CO INC (US) 2002-11-20 EP claimed
EP-0925302-A1 PALLADIUM CATALYZED INDOLIZATION Merck & Co., Inc. (US) 1999-06-30 EP claimed
US-5808064-A HYDROSILATION OF AN INDOLE AS CHEMICAL INTERMEDIATE MERCK & CO., INC. (US) 1998-09-15 US claimed
WO-1998006725-A1 PALLADIUM CATALYZED INDOLIZATION MERCK & CO., INC. (US) 1998-02-19 WO claimed
US-5567824-A CATALYZING THE CYCLIZATION IN PRESENCE OF A SOLVENT AND A PROTON ACCEPTOR MERCK & CO., INC. (US) 1996-10-22 US claimed
EP-0763032-B1 PALLADIUM CATALYZED RING CLOSURE OF TRIAZOLYL TRYPTAMINE MERCK & CO INC (US) 2003-10-15 EP disclosed
EP-0925302-B1 PALLADIUM CATALYZED INDOLIZATION MERCK & CO INC (US) 2002-11-20 EP disclosed
US-5808064-A HYDROSILATION OF AN INDOLE AS CHEMICAL INTERMEDIATE MERCK & CO., INC. (US) 1998-09-15 US disclosed
US-5567824-A CATALYZING THE CYCLIZATION IN PRESENCE OF A SOLVENT AND A PROTON ACCEPTOR MERCK & CO., INC. (US) 1996-10-22 US disclosed