SCHEMBL6946595

SCHEMBL6946595

CCOC(=O)OC1CC(c2ccccc2Cl)c2c(Cl)cc(Cl)cc2N1

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.41
TSHR P16473 1/20 0.41
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
ALOX12 P18054 1/20 0.39
CYP2C19 P33261 1/20 0.39
MAPK1 P28482 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6949286 0.93 CA1 (0.37) POLBTSHRMAPK1
SCHEMBL6952854 0.91 ALDH1A1 (0.36) POLBTSHR
SCHEMBL6951131 0.91 POLB (0.35) POLBTSHRMAPK1
SCHEMBL6951129 0.89 MEN1 (0.39) CYP3A4CYP2C19
SCHEMBL6946932 0.86 MAPK1 (0.37) CYP3A4MAPK1
SCHEMBL6948161 0.86 NPSR1 (0.38) POLBCYP3A4CYP2C9CYP2C19MAPK1
SCHEMBL7546562 0.85 ABCC1 (0.38) ALOX12MAPK1
SCHEMBL6640286 0.85 MEN1 (0.42) CYP3A4CYP2C19
SCHEMBL6947977 0.85 MAPK1 (0.38) MAPK1
SCHEMBL6945541 0.84 MAPK1 (0.35) MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2003522758-A 2003-07-29 JP claimed
EP-1254118-A2 SUBSTITUTED 1,2,3,4- TETRAHYDROQUINOLINE-2-CARBOXYLIC ACID DERIVATIVES Grünenthal GmbH (DE) 2002-11-06 EP claimed
WO-2001058875-A2 SUBSTITUTED 1,2,3,4- TETRAHYDROQUINOLINE-2-CARBOXYLIC ACID DERIVATIVES Grünenthal GmbH (DE) 2001-08-16 WO claimed
EP-1254118-A2 SUBSTITUTED 1,2,3,4- TETRAHYDROQUINOLINE-2-CARBOXYLIC ACID DERIVATIVES Grünenthal GmbH (DE) 2002-11-06 EP disclosed
WO-2001058875-A2 SUBSTITUTED 1,2,3,4- TETRAHYDROQUINOLINE-2-CARBOXYLIC ACID DERIVATIVES Grünenthal GmbH (DE) 2001-08-16 WO disclosed