SCHEMBL7546562

SCHEMBL7546562

CCOC(=O)OC1CC(c2ccc(Cl)cc2)c2c(Cl)cc(Cl)cc2N1

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ABCC1 P33527 1/20 0.38
ALOX12 P18054 2/20 0.38
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38
MAPK1 P28482 1/20 0.38
GAA P10253 2/20 0.37
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6945541 0.95 MAPK1 (0.35) MAPK1
SCHEMBL6952784 0.93 GAA (0.35) GAA
SCHEMBL6952693 0.93 MAPT (0.35) LMNAHTTALDH1A1
SCHEMBL6951129 0.93 MEN1 (0.39)
SCHEMBL7489535 0.91 CYP2D6 (0.36) MAPK1
SCHEMBL6947134 0.89 ALDH1A1 (0.38) MAPK1ALDH1A1
SCHEMBL6947977 0.89 MAPK1 (0.38) LMNAMAPK1
SCHEMBL6946334 0.88 MMP13 (0.36)
SCHEMBL6949316 0.86 ALDH1A1 (0.35) MAPK1ALDH1A1
SCHEMBL6944762 0.86 ALDH1A1 (0.37) LMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1254118-A2 SUBSTITUTED 1,2,3,4- TETRAHYDROQUINOLINE-2-CARBOXYLIC ACID DERIVATIVES Grünenthal GmbH (DE) 2002-11-06 EP disclosed
WO-2001058875-A2 SUBSTITUTED 1,2,3,4- TETRAHYDROQUINOLINE-2-CARBOXYLIC ACID DERIVATIVES Grünenthal GmbH (DE) 2001-08-16 WO disclosed