SCHEMBL6946616

SCHEMBL6946616

CCCCCCCCCC(=O)OCN1C(=O)C(c2cn(C)c3ccccc23)=C(c2cn(C)c3cc([N+](=O)[O-])ccc23)C1=O

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 4/20 0.45
CDK9 P50750 4/20 0.45
CDK2 P24941 2/20 0.45
CCNA2 P20248 1/20 0.45
MAPT P10636 1/20 0.41
PRKCA P17252 1/20 0.40
PRKCE Q02156 1/20 0.40
RASGRP3 Q8IV61 1/20 0.40
ALDH1A1 P00352 1/20 0.39
TDP1 Q9NUW8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6955491 0.95 CCNT1 (0.42) CCNT1CDK9CDK2CCNA2MAPT
SCHEMBL6956384 0.92 CCNT1 (0.46) CCNT1CDK9CDK2CCNA2
SCHEMBL7164524 0.89 CCNT1 (0.47) CCNT1CDK9CDK2CCNA2
SCHEMBL7500940 0.86 CCNT1 (0.46) CCNT1CDK9CDK2CCNA2
SCHEMBL6947835 0.84 CCNT1 (0.44) CCNT1CDK9CDK2CCNA2MAPT
SCHEMBL7508601 0.83 CCNT1 (0.47) CCNT1CDK9CDK2CCNA2
SCHEMBL6956508 0.83 CCNT1 (0.42) CCNT1CDK9CDK2CCNA2ALDH1A1
SCHEMBL6954175 0.82 CCNT1 (0.43) CCNT1CDK9CDK2CCNA2RASGRP3
SCHEMBL6954265 0.82 CDK9 (0.39) CCNT1CDK9CDK2CCNA2PRKCA
Hydrochloric Acid SCHEMBL6954170 0.81 CCNT1 (0.42) CCNT1CDK9CDK2CCNA2RASGRP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1155595-C Substituted pyrroles as antiproliferative agents for the treatment of cancer - 2004-06-30 CN claimed
EP-1224181-B1 SUBSTITUTED PYRROLES AS ANTIPROLIFERATIVE AGENTS FOR THE TREATMENT OF CANCER HOFFMANN LA ROCHE (CH) 2003-12-03 EP claimed
CN-1378545-A Substituted pyrroles as antiproliferative agents for treatment of cancer HOFFMANN LA ROCHE (CH) 2002-11-06 CN claimed
CN-1155595-C Substituted pyrroles as antiproliferative agents for the treatment of cancer - 2004-06-30 CN disclosed
CN-1378545-A Substituted pyrroles as antiproliferative agents for treatment of cancer HOFFMANN LA ROCHE (CH) 2002-11-06 CN disclosed