SCHEMBL6947064

SCHEMBL6947064

O=C(O)CNC(=O)[C@@H](O)C(Cc1ccccc1)NC(=O)c1cccc(NS(=O)(=O)c2ccc3ccccc3c2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSD P07339 2/20 0.48
BACE1 P56817 2/20 0.48
BACE2 Q9Y5Z0 1/20 0.48
AKR1C3 P42330 1/20 0.47
CCR1 P32246 1/20 0.44
GGPS1 O95749 1/20 0.44
F2 P00734 2/20 0.43
GPR27 Q9NS67 1/20 0.43
SLC16A3 O15427 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
HTT P42858 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
ALDH1A1 P00352 2/20 0.41
OPRM1 P35372 1/20 0.41
OPRD1 P41143 1/20 0.41
POLB P06746 1/20 0.41
MAPT P10636 1/20 0.41
PFKFB3 Q16875 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6939930 0.90 AR (0.48) CTSDBACE1BACE2AKR1C3CCR1
SCHEMBL7309549 0.89 AKR1C3 (0.52) CTSDBACE1BACE2AKR1C3CCR1
SCHEMBL7322714 0.88 AKR1C3 (0.51) CTSDBACE1BACE2AKR1C3CCR1
SCHEMBL7325408 0.84 AR (0.52) CTSDBACE1BACE2AKR1C3CCR1
SCHEMBL6944325 0.83 AKR1C3 (0.48) AKR1C3GGPS1F2GPR27SLC16A3
SCHEMBL6942392 0.83 AKR1C3 (0.48) AKR1C3GGPS1F2GPR27SLC16A3
SCHEMBL7791333 0.80 AKR1C3 (0.54) AKR1C3GGPS1F2GPR27SLC16A3
SCHEMBL7791335 0.80 AKR1C3 (0.54) AKR1C3GGPS1F2GPR27SLC16A3
SCHEMBL7782218 0.79 AKR1C3 (0.53) AKR1C3GGPS1F2GPR27SLC16A3
SCHEMBL7782219 0.79 AKR1C3 (0.53) AKR1C3GGPS1F2GPR27SLC16A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0944582-B1 KETOBENZAMIDES AS CALPAIN INHIBITORS ABBOTT GMBH & CO KG (DE) 2003-07-02 EP disclosed
US-6103720-A ENZYME INHIBITORS; ANTIICHEMIC AND -TUMOR AGENTS; STROKES; ALZEIMER'S DISEASE BASF AKTIENGESELLSCHAFT (DE) 2000-08-15 US disclosed
EP-0944582-A1 KETOBENZAMIDES AS CALPAIN INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1999-09-29 EP disclosed
WO-1998025883-A1 KETOBENZAMIDES AS CALPAIN INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1998-06-18 WO disclosed