SCHEMBL7325408

SCHEMBL7325408

CCOC(=O)[C@@H](O)C(Cc1ccccc1)NC(=O)c1cccc(NS(=O)(=O)c2ccc3ccccc3c2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.52
CTSD P07339 1/20 0.48
BACE1 P56817 1/20 0.48
BACE2 Q9Y5Z0 1/20 0.48
AKR1C3 P42330 1/20 0.47
KAT6A Q92794 4/20 0.46
HIF1A Q16665 1/20 0.45
OPRM1 P35372 1/20 0.45
OPRD1 P41143 1/20 0.45
PLG P00747 1/20 0.45
LMNA P02545 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
CCR1 P32246 1/20 0.44
GGPS1 O95749 1/20 0.44
PLAU P00749 1/20 0.44
F2 P00734 1/20 0.43
GPR27 Q9NS67 1/20 0.43
ALDH1A1 P00352 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6939930 0.90 AR (0.48) ARCTSDBACE1BACE2AKR1C3
SCHEMBL7309549 0.89 AKR1C3 (0.52) CTSDBACE1BACE2AKR1C3KAT6A
SCHEMBL7322714 0.88 AKR1C3 (0.51) ARCTSDBACE1BACE2AKR1C3
SCHEMBL6947064 0.84 CTSD (0.48) ARCTSDBACE1BACE2AKR1C3
SCHEMBL7791333 0.80 AKR1C3 (0.54) ARAKR1C3KAT6ALMNASMN1; SMN2
SCHEMBL7791335 0.80 AKR1C3 (0.54) ARAKR1C3KAT6ALMNASMN1; SMN2
SCHEMBL6942097 0.79 CAPN1 (0.53) AKR1C3KAT6APLGGGPS1PLAU
SCHEMBL7313713 0.79 CAPN1 (0.53) AKR1C3KAT6APLGGGPS1PLAU
SCHEMBL7782218 0.79 AKR1C3 (0.53) ARAKR1C3KAT6ALMNASMN1; SMN2
SCHEMBL7782219 0.79 AKR1C3 (0.53) ARAKR1C3KAT6ALMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6103720-A ENZYME INHIBITORS; ANTIICHEMIC AND -TUMOR AGENTS; STROKES; ALZEIMER'S DISEASE BASF AKTIENGESELLSCHAFT (DE) 2000-08-15 US disclosed