SCHEMBL6947201

SCHEMBL6947201

OC1CCCc2cc(F)cc(F)c21

nearest known ligand 0.38

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 4/20 0.33
UGT2B17 O75795 2/20 0.33
EPAS1 Q99814 2/20 0.32
CYP11B1 P15538 2/20 0.31
CYP11B2 P19099 2/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL326748 0.89 CYP11B1 (0.38) EPAS1CYP11B1CYP11B2
SCHEMBL13612885 0.82 UGT2B17 (0.31) HTR6UGT2B17CYP11B1CYP11B2
SCHEMBL31127749 0.82 EPAS1 (0.32) UGT2B17EPAS1
SCHEMBL27982324 0.74 HTR6 (0.33) HTR6
SCHEMBL29197997 0.74
SCHEMBL30858742 0.72 HTR6 (0.36) HTR6RAB9A
SCHEMBL24593689 0.70 UGT2B17 (0.51) UGT2B17EPAS1CYP11B1CYP11B2
SCHEMBL6958845 0.70 UGT2B17 (0.51) UGT2B17EPAS1CYP11B1CYP11B2
SCHEMBL16800617 0.70 CYP11B1 (0.37) CYP11B1CYP11B2
SCHEMBL13882545 0.70 PGR (0.45) HTR6UGT2B17CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0757677-B1 BENZOCYCLOHEXYLIMIDAZOLETHIONE DERIVATIVES SYNTEX LLC (US) 2003-06-18 EP disclosed
US-5719280-A REACTING AMINE SUBSTITUTED BENZOCYCLOALKANE WITH DIALKYLOXYACETALDEHYDE IN PRESENCE OF REDUCING AGENT OR CATALYTIC HYDROGENATION, TREATING WITH THIOCYANIC ACID SYNTEX (U.S.A.) INC. (US) 1998-02-17 US disclosed
EP-0757677-A1 BENZOCYCLOALKYLAZOLETHIONE DERIVATIVES SYNTEX (U.S.A.) INC. (US) 1997-02-12 EP disclosed
US-5538988-A CARDIOVASCULAR DISORDERS AND DOPAMINE HYDROLASE ENZYME INHIBITORS SYNTEX (U.S.A.) INC. 1996-07-23 US disclosed
WO-1995029165-A2 BENZOCYCLOALKYLAZ0LETHIONE DERIVATIVES AS DOPAMIN BETA-HYDROXYLASE INHIBITORS SYNTEX (U.S.A.) INC. (US) 1995-11-02 WO disclosed