SCHEMBL6947485

SCHEMBL6947485

CCCCNCCCC.CCCN1CCC(=O)CC1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.38
ALDH1A1 P00352 3/20 0.37
TSHR P16473 2/20 0.37
CYP1A2 P05177 1/20 0.36
THRB P10828 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
GNAI3 P08754 1/20 0.35
GNAO1 P09471 1/20 0.35
GNAI1 P63096 1/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 1/20 0.35
RXFP1 Q9HBX9 1/20 0.34
ACE2 Q9BYF1 1/20 0.34
GAA P10253 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7246872 0.93 ACE2 (0.42) ALDH1A1TSHRCYP1A2THRBL3MBTL1
SCHEMBL6947718 0.93 ALDH1A1 (0.39) ALDH1A1TSHRCYP1A2THRBL3MBTL1
SCHEMBL6945104 0.91 GNAI3 (0.41) ALDH1A1TSHRGNAI3GNAO1GNAI1
SCHEMBL6947802 0.89 POLB (0.40) POLBALDH1A1CYP1A2THRBL3MBTL1
SCHEMBL6943645 0.87 ALDH1A1 (0.40) POLBALDH1A1TSHRCYP1A2THRB
SCHEMBL6948499 0.86 ALDH1A1 (0.39) ALDH1A1THRBL3MBTL1GNAI3GNAO1
SCHEMBL8114400 0.84 POLB (0.46) POLBALDH1A1THRBL3MBTL1NPC1
SCHEMBL1180845 0.84 POLB (0.46) POLBALDH1A1THRBL3MBTL1NPC1
SCHEMBL6942247 0.84 GNAI3 (0.41) GNAI3GNAO1GNAI1GAA
Diethylamine SCHEMBL6947450 0.83 POLB (0.41) POLBALDH1A1CYP1A2THRBL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6642231-B2 Antineoplastic agents, treatment for neuronal injury and degeneration AVENTIS PHARMACEUTICALS INC. 2003-11-04 US disclosed
EP-1056744-B1 6,9-DISUBSTITUTED 2- TRANS-(4- AMINOCYCLOHEXYL) AMINO]PURINES AVENTIS PHARMA INC (US) 2003-10-22 EP disclosed
US-20030105098-A1 6,9-disubstituted 2-[trans-(4-aminocyclohexyl) amino] purines AVENTISUB II INC. 2003-06-05 US disclosed
US-6479487-B1 INHIBIT CYCLIN DEPENDENT KINASES, PARTICULARLY CDK-2; ANTIAPOPTOSIS AGENT; INHIBITS DEVELOPMENT OF NEOPLASMS AVENTIS PHARMACEUTICALS INC. 2002-11-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030105098-A1 6,9-disubstituted 2-[trans-(4-aminocyclohexyl) amino] purines CDK6, CDK5, CDK2 POLB 413/4885ALDH1A1 2147/4885TSHR 4411/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.