SCHEMBL6947809

SCHEMBL6947809

O=C(O)/C(O)=C/C(=O)c1cc(O)cc(OCc2ccccc2)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.56
KMT2A Q03164 1/20 0.56
NR4A2 P43354 2/20 0.50
CYP1A2 P05177 2/20 0.50
CYP1A1 P04798 1/20 0.50
CYP19A1 P11511 1/20 0.50
MAOB P27338 3/20 0.48
PTPN1 P18031 1/20 0.47
NR4A1 P22736 1/20 0.47
NR4A3 Q92570 1/20 0.47
SLC5A1 P13866 1/20 0.46
SLC5A2 P31639 1/20 0.46
SMPD1 P17405 1/20 0.46
ABCG2 Q9UNQ0 1/20 0.45
SRD5A2 P31213 2/20 0.45
PARP10 Q53GL7 1/20 0.44
GSK3B P49841 2/20 0.44
BACE1 P56817 2/20 0.44
GPBAR1 Q8TDU6 1/20 0.44
LMNA P02545 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6947812 1.00 MEN1 (0.56) MEN1KMT2ANR4A2CYP1A2CYP1A1
SCHEMBL6947862 0.93 MEN1 (0.65) MEN1KMT2ANR4A2MAOBPTPN1
SCHEMBL6947866 0.93 MEN1 (0.65) MEN1KMT2ANR4A2MAOBPTPN1
SCHEMBL6947101 0.87 MEN1 (0.57) MEN1KMT2ANR4A2MAOBPTPN1
SCHEMBL6947103 0.87 MEN1 (0.57) MEN1KMT2ANR4A2MAOBPTPN1
SCHEMBL6950489 0.85 NR4A2 (0.67) MEN1KMT2ANR4A2MAOBPTPN1
SCHEMBL6950492 0.85 NR4A2 (0.67) MEN1KMT2ANR4A2MAOBPTPN1
SCHEMBL14259572 0.84 MAOB (0.55) MEN1KMT2ANR4A2MAOBPTPN1
SCHEMBL3888880 0.83 NR4A1 (0.64) NR4A2CYP1A2MAOBPTPN1NR4A1
SCHEMBL3888888 0.83 NR4A1 (0.64) NR4A2CYP1A2MAOBPTPN1NR4A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP claimed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP claimed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO claimed
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP disclosed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US disclosed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP disclosed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO disclosed