SCHEMBL6950489

SCHEMBL6950489

O=C(O)/C(O)=C/C(=O)c1cccc(OCc2ccccc2)c1

nearest known ligand 0.67

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 6/20 0.67
MAOB P27338 2/20 0.63
PTPN1 P18031 1/20 0.61
SMPD1 P17405 2/20 0.60
SRD5A2 P31213 1/20 0.59
MEN1 O00255 1/20 0.54
KMT2A Q03164 1/20 0.54
NR1H4 Q96RI1 1/20 0.53
ALDH1A1 P00352 2/20 0.52
KDM4E B2RXH2 1/20 0.52
PKM P14618 1/20 0.52
MRGPRX4 Q96LA9 1/20 0.52
GPR132 Q9UNW8 1/20 0.52
MAOA P21397 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6950492 1.00 NR4A2 (0.67) NR4A2MAOBPTPN1SMPD1SRD5A2
SCHEMBL6940936 0.90 NR4A2 (0.70) NR4A2MAOBPTPN1SMPD1MEN1
SCHEMBL6940932 0.90 NR4A2 (0.70) NR4A2MAOBPTPN1SMPD1MEN1
SCHEMBL6946121 0.90 MAOB (0.66) NR4A2MAOBPTPN1SMPD1NR1H4
SCHEMBL6946117 0.90 MAOB (0.66) NR4A2MAOBPTPN1SMPD1NR1H4
SCHEMBL6951859 0.90 NR4A2 (0.70) NR4A2MAOBPTPN1MEN1KMT2A
SCHEMBL6951854 0.90 NR4A2 (0.70) NR4A2MAOBPTPN1MEN1KMT2A
SCHEMBL6947866 0.89 MEN1 (0.65) NR4A2MAOBPTPN1SMPD1SRD5A2
SCHEMBL6947862 0.89 MEN1 (0.65) NR4A2MAOBPTPN1SMPD1SRD5A2
SCHEMBL6205727 0.89 MRGPRX4 (0.63) NR4A2MAOBPTPN1SMPD1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP disclosed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US disclosed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP disclosed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO disclosed