SCHEMBL6948018

SCHEMBL6948018

CC(C)Oc1ccc(Cc2ccccc2)cc1C#N

nearest known ligand 0.45

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
XDH P47989 4/20 0.45
MAOB P27338 1/20 0.43
S1PR1 P21453 6/20 0.42
S1PR5 Q9H228 2/20 0.42
NPY2R P49146 1/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8799523 0.81 XDH (0.46) XDHS1PR1S1PR5
SCHEMBL932494 0.80 S1PR1 (0.47) XDHS1PR1S1PR5
SCHEMBL31470411 0.80 XDH (0.45) XDHS1PR1S1PR5
SCHEMBL1919413 0.80 XDH (0.48) XDHS1PR1S1PR5
SCHEMBL31185537 0.80 XDH (0.48) XDHS1PR1S1PR5
SCHEMBL26179844 0.79 S1PR1 (0.46) XDHS1PR1S1PR5
Dimethylamine SCHEMBL6948153 0.78 MAOB (0.46) XDHMAOBNPY2R
SCHEMBL20057756 0.77 XDH (0.42) XDHS1PR1S1PR5
SCHEMBL28531441 0.75 XDH (0.44) XDHS1PR1S1PR5NPY2R
SCHEMBL6948151 0.75 LTA4H (0.57) MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP disclosed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US disclosed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP disclosed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO disclosed