SCHEMBL6948023

SCHEMBL6948023

O=CCc1cccc(Sc2ccccc2)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 2/20 0.58
HTR6 P50406 1/20 0.58
SLC6A4 P31645 1/20 0.41
MAOB P27338 3/20 0.40
MAOA P21397 2/20 0.40
BCL2 P10415 1/20 0.38
MCL1 Q07820 1/20 0.38
HPGD P15428 3/20 0.36
ALDH1A1 P00352 2/20 0.36
LMNA P02545 2/20 0.36
SIRT1 Q96EB6 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ADH1B P00325 1/20 0.35
ADH1C P00326 1/20 0.35
ADH1A P07327 1/20 0.35
ADH7 P40394 1/20 0.35
ANXA2 P07355 1/20 0.35
S100A10 P60903 1/20 0.35
KMT2A Q03164 1/20 0.35
ATM Q13315 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3825516 0.82 SLC6A4 (0.48) HTR2CHTR6SLC6A4MAOBMAOA
SCHEMBL14051500 0.82 HPGD (0.41) HTR2CHTR6MAOBMAOAHPGD
SCHEMBL1295549 0.78 MAPT (0.43) HPGDALDH1A1SMN1; SMN2KMT2APOLB
SCHEMBL20126552 0.78 HTR2C (0.63) HTR2CHTR6SLC6A4MAOBMAOA
SCHEMBL12345478 0.76 MAOB (0.39) MAOBMAOALMNAADH1BADH1C
SCHEMBL920219 0.76 HTR6 (0.72) HTR2CHTR6SLC6A4MAOBMAOA
SCHEMBL1680382 0.76 HTR2C (0.61) HTR2CHTR6SLC6A4MAOBMAOA
SCHEMBL8783743 0.76 AKR1B1 (0.57) HTR2CHTR6HPGDALDH1A1LMNA
SCHEMBL1295715 0.74 FFAR4 (0.42) ALDH1A1LMNAATM
SCHEMBL13377220 0.74 MAOB (0.52) MAOBMAOAHPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP disclosed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP disclosed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO disclosed