SCHEMBL6948113

SCHEMBL6948113

COCCOc1c(Br)cc(-c2ccccc2)cc1OC

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 8/20 0.45
L3MBTL1 Q9Y468 6/20 0.45
LMNA P02545 4/20 0.45
MIF P14174 1/20 0.44
SMN1; SMN2 Q16637 3/20 0.41
RAB9A P51151 1/20 0.41
ALDH1A1 P00352 4/20 0.41
FYN P06241 1/20 0.41
HPGD P15428 4/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
KDM4E B2RXH2 3/20 0.40
GAA P10253 1/20 0.40
THRB P10828 1/20 0.40
BLM P54132 1/20 0.40
HTT P42858 1/20 0.40
TDP1 Q9NUW8 2/20 0.39
MAPK1 P28482 1/20 0.39
ALOX15 P16050 1/20 0.39
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6946141 0.80 KMT2A (0.49) MAPTL3MBTL1LMNASMN1; SMN2ALDH1A1
SCHEMBL6946935 0.77 CNR2 (0.47) MAPTL3MBTL1LMNASMN1; SMN2RAB9A
SCHEMBL29260702 0.75 MGAM (0.41) MAPTL3MBTL1SMN1; SMN2RAB9AALDH1A1
Methoxy Aucuparin SCHEMBL8420787 0.73 KDM4E (0.62) MAPTL3MBTL1SMN1; SMN2ALDH1A1FYN
SCHEMBL6943688 0.72 ALDH1A1 (0.64) MAPTL3MBTL1LMNASMN1; SMN2RAB9A
SCHEMBL28338665 0.71 HPGD (0.61) MAPTL3MBTL1LMNASMN1; SMN2ALDH1A1
SCHEMBL7169549 0.69 IKBKB (0.48) SMN1; SMN2RAB9AALDH1A1FYNKDM4E
Biphenyl SCHEMBL4856272 0.69 ALDH1A1 (0.50) LMNAALDH1A1HPGDKDM4ETDP1
SCHEMBL3924409 0.69 MAPT (0.57) MAPTL3MBTL1LMNASMN1; SMN2RAB9A
SCHEMBL456627 0.69 ABCG2 (0.47) MAPTL3MBTL1RAB9AALDH1A1FYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP disclosed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP disclosed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO disclosed