SCHEMBL6948968

SCHEMBL6948968

Nc1nc(CCOc2ccccc2)c2nc[nH]c2n1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DHFR P00374 11/20 0.46
CDK1 P06493 1/20 0.42
CCNB1 P14635 1/20 0.42
CCNA2 P20248 1/20 0.42
CDK2 P24941 1/20 0.42
CCNA1 P78396 1/20 0.42
NPC1 O15118 3/20 0.41
RAB9A P51151 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HRH3 Q9Y5N1 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.38
MPO P05164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL821881 0.82 CDK1 (0.46) DHFRCDK1CCNB1CCNA2CDK2
SCHEMBL6950876 0.82 MPO (0.56) DHFRCDK1CCNB1CCNA2CDK2
SCHEMBL6946759 0.80 CYP2D6 (0.48) DHFRCDK1CCNB1CCNA2CDK2
SCHEMBL6948069 0.80 MPO (0.47) DHFRCDK1CCNB1CCNA2CDK2
SCHEMBL12227593 0.79 CDK1 (0.43) DHFRCDK1CCNB1CCNA2CDK2
Hydrochloric Acid SCHEMBL5731125 0.75 TLR7 (0.35) DHFRL3MBTL1
SCHEMBL9681378 0.74 TRPA1 (0.43) CDK1CCNB1CCNA2CDK2CCNA1
SCHEMBL10743106 0.73 JAK2 (0.46) CDK1CCNB1CCNA2CDK2CCNA1
SCHEMBL7527092 0.72 CDK1 (0.31) CDK1CCNB1CCNA2CDK2CCNA1
SCHEMBL6950562 0.71 CDK1 (0.42) CDK1CCNB1CCNA2CDK2CCNA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1349857-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2003-10-08 EP disclosed
WO-2002055521-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2002-07-18 WO disclosed