SCHEMBL6949154

SCHEMBL6949154

CC(C)(C)OC(=O)ON1CC(O)C(c2ccc(Br)cc2)C(COC(c2ccccc2)(c2ccccc2)c2ccccc2)C1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RORC P51449 4/20 0.38
ALDH1A1 P00352 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
GAA P10253 1/20 0.32
CYP2D6 P10635 1/20 0.32
MAPT P10636 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
HTT P42858 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
SLC6A1 P30531 3/20 0.31
SLC6A11 P48066 1/20 0.31
NR1H2 P55055 1/20 0.30
NR1H3 Q13133 1/20 0.30
HDAC4 P56524 1/20 0.30
BCL2 P10415 1/20 0.30
BECN1 Q14457 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6956483 0.88 MAPT (0.35) RORCALDH1A1CYP1A2CYP3A4GAA
SCHEMBL6959407 0.88 HDAC1 (0.34) ALDH1A1CYP3A4MAPTSLC6A1SLC6A11
SCHEMBL6953593 0.83 REN (0.39) ALDH1A1GAAL3MBTL1
SCHEMBL6948019 0.83 RORC (0.36) RORCALDH1A1CYP1A2CYP3A4GAA
SCHEMBL7076803 0.82 REN (0.39) MAPT
SCHEMBL6959116 0.81 RORC (0.35) RORCNR1H2NR1H3
SCHEMBL6044052 0.80 MAPT (0.38) RORCALDH1A1CYP1A2CYP3A4GAA
SCHEMBL6954547 0.75 PLA2G10 (0.37) RORC
SCHEMBL7081784 0.74 REN (0.39)
SCHEMBL7082373 0.74 REN (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863875-B1 NEW 4-(OXYALKOXYPHENYL)-3-OXY-PIPERIDINES FOR TREATING HEART AND KIDNEY INSUFFICIENCY HOFFMANN LA ROCHE (CH) 2003-06-04 EP disclosed
EP-0863875-A1 NEW 4-(OXYALKOXYPHENYL)-3-OXY-PIPERIDINES FOR TREATING HEART AND KIDNEY INSUFFICIENCY F. HOFFMANN-LA ROCHE AG (CH) 1998-09-16 EP disclosed
WO-1997009311-A1 NEW 4-(OXYALKOXYPHENYL)-3-OXY-PIPERIDINES FOR TREATING HEART AND KIDNEY INSUFFICIENCY F. HOFFMANN-LA ROCHE AG (CH) 1997-03-13 WO disclosed