SCHEMBL6949840

SCHEMBL6949840

O=C(O)C(O)=CC(=O)c1ccc2[nH]c(Cc3ccc(F)cc3)cc2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F2 P00734 4/20 0.47
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 2/20 0.37
HPGD P15428 2/20 0.37
PDPK1 O15530 1/20 0.37
LMNA P02545 1/20 0.37
TSHR P16473 1/20 0.37
NFKB1 P19838 1/20 0.37
APEX1 P27695 1/20 0.37
CYP2C19 P33261 1/20 0.37
HSD17B10 Q99714 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
CTNNB1 P35222 1/20 0.37
WNT3A P56704 1/20 0.37
FFAR1 O14842 2/20 0.36
PPARG P37231 1/20 0.36
PIN1 Q13526 1/20 0.36
GPER1 Q99527 1/20 0.36
DAO P14920 2/20 0.35
FLT3 P36888 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6950558 0.92 ITK (0.39) F2KDM4EALDH1A1HPGDLMNA
SCHEMBL27926719 0.78 F2 (0.48) F2KDM4EALDH1A1HPGDPDPK1
SCHEMBL4675001 0.77 ALDH1A1 (0.38) KDM4EALDH1A1HPGDLMNADAO
SCHEMBL4675004 0.77 ALDH1A1 (0.38) KDM4EALDH1A1HPGDLMNADAO
SCHEMBL6946214 0.76 BRS3 (0.36) KDM4EHSD17B10PPARGDAO
Hydroxyamine SCHEMBL4796191 0.74 NR4A2 (0.46) F2KDM4EALDH1A1HPGDAPEX1
SCHEMBL4670507 0.74 DAO (0.36) KDM4EALDH1A1HPGDLMNADAO
SCHEMBL4670505 0.74 DAO (0.36) KDM4EALDH1A1HPGDLMNADAO
SCHEMBL977626 0.72 F2 (0.70) F2KDM4EALDH1A1HPGDTSHR
SCHEMBL8105255 0.72 MAPT (0.58) KDM4EALDH1A1HPGDCYP2C19MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP claimed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP claimed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO claimed
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP disclosed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP disclosed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO disclosed