SCHEMBL6950436

SCHEMBL6950436

COCCN(C)C(=O)Nc1c(C(=O)c2ccccc2)[nH]c2cc(Cl)ccc12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
NPC1 O15118 1/20 0.41
ALDH1A1 P00352 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
HPGD P15428 1/20 0.41
ALOX12 P18054 1/20 0.41
RAB9A P51151 1/20 0.41
KMT2A Q03164 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
TP53 P04637 1/20 0.41
MCL1 Q07820 5/20 0.40
MDM2 Q00987 1/20 0.40
CNR1 P21554 1/20 0.39
TUBB4A P04350 1/20 0.39
TUBB P07437 1/20 0.39
TUBA3C P0DPH7 1/20 0.39
TUBA1B P68363 1/20 0.39
TUBA4A P68366 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6954387 0.89 CNR1 (0.41) TP53CNR1ALOX15
SCHEMBL6954712 0.87 CNR1 (0.42) KDM4EMEN1NPC1ALDH1A1GAA
SCHEMBL6951194 0.85 RAB9A (0.44) KDM4EMEN1NPC1ALDH1A1GAA
SCHEMBL6954685 0.85 MEN1 (0.43) KDM4EMEN1NPC1ALDH1A1GAA
SCHEMBL6950527 0.84 MEN1 (0.42) KDM4EMEN1NPC1ALDH1A1GAA
SCHEMBL6951362 0.82 CNR1 (0.44) KDM4EMEN1NPC1ALDH1A1GAA
SCHEMBL6948046 0.82 CNR1 (0.43) KDM4EMEN1NPC1ALDH1A1GAA
SCHEMBL7506712 0.82 KDM4E (0.53) KDM4EMEN1NPC1ALDH1A1GAA
SCHEMBL6946118 0.81 ALDH1A1 (0.54) KDM4EMEN1NPC1ALDH1A1GAA
SCHEMBL7502892 0.80 SERPINE1 (0.48) KDM4EMEN1NPC1ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0985666-B1 Substituted indole compounds as COX-2 inhibitors PFIZER (US) 2003-11-05 EP claimed
US-6277878-B1 ANTIINFLAMMATORY AGENTS; ANALGESICS PFIZER INC 2001-08-21 US claimed
EP-0985666-A1 Substituted indole compounds as COX-2 inhibitors PFIZER INC. (US) 2000-03-15 EP claimed
EP-0985666-B1 Substituted indole compounds as COX-2 inhibitors PFIZER (US) 2003-11-05 EP disclosed
US-6277878-B1 ANTIINFLAMMATORY AGENTS; ANALGESICS PFIZER INC 2001-08-21 US disclosed
EP-0985666-A1 Substituted indole compounds as COX-2 inhibitors PFIZER INC. (US) 2000-03-15 EP disclosed