SCHEMBL695189

SCHEMBL695189

COC(=O)C1C[C@@H](S(=O)(=O)c2ccccc2Cl)CN1c1cc(C)nn1-c1ccc(C(F)(F)F)cc1

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CTSS P25774 16/20 0.49
ELOVL6 Q9H5J4 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.41
CTSL P07711 5/20 0.39
CTSB P07858 4/20 0.39
CTSK P43235 2/20 0.38
CRHR1 P34998 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2104910 1.00 CTSS (0.49) CTSSELOVL6SMN1; SMN2CTSLCTSB
SCHEMBL696030 0.91 CTSS (0.45) CTSSELOVL6CTSLCTSBCTSK
SCHEMBL694697 0.90 ELOVL6 (0.41) CTSSELOVL6SMN1; SMN2CTSLCTSB
SCHEMBL2105211 0.90 ELOVL6 (0.41) CTSSELOVL6SMN1; SMN2CTSLCTSB
SCHEMBL2105284 0.87 SMN1; SMN2 (0.41) CTSSSMN1; SMN2CTSLCTSBCTSK
SCHEMBL696422 0.87 SMN1; SMN2 (0.41) CTSSSMN1; SMN2CTSLCTSBCTSK
SCHEMBL697407 0.86 CTSS (0.52) CTSSSMN1; SMN2CTSLCTSBCTSK
SCHEMBL2105017 0.86 CTSS (0.52) CTSSSMN1; SMN2CTSLCTSBCTSK
SCHEMBL695699 0.85 CTSS (0.58) CTSSCTSLCTSB
SCHEMBL694847 0.84 CTSS (0.49) CTSSCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2421826-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. Hoffmann-La Roche AG (CH) 2012-02-29 EP disclosed
WO-2010121918-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2010-10-28 WO disclosed