SCHEMBL6954402

SCHEMBL6954402

Cc1ccc(S(=O)(=O)SCc2cccc(-c3cc4ccccc4o3)c2)cc1

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BCHE P06276 9/20 0.56
ACHE P22303 9/20 0.56
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
RXFP1 Q9HBX9 1/20 0.47
CA9 Q16790 2/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
P2RY14 Q15391 1/20 0.45
MAOB P27338 2/20 0.44
MAOA P21397 1/20 0.44
PTGES2 Q9H7Z7 1/20 0.42
CA12 O43570 1/20 0.42
PSMB5 P28074 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8434487 0.74 BCHE (0.76) BCHEACHE
SCHEMBL11607679 0.74 BCHE (1.00) BCHEACHEALDH1A1CA9CA12
SCHEMBL4911544 0.71 CA9 (0.54) KDM4EALDH1A1NPSR1RXFP1CA9
SCHEMBL13140660 0.71 MAOB (0.65) KDM4EALDH1A1CA9CA1CA2
SCHEMBL3687533 0.71 MAOB (0.68) KDM4EALDH1A1CA9CA1CA2
SCHEMBL6959012 0.69 BCHE (0.71) BCHEACHEALDH1A1
SCHEMBL6959190 0.69 BCHE (0.83) BCHEACHEALDH1A1CA9CA1
SCHEMBL8434517 0.69 BCHE (0.72) BCHEACHEMAOB
SCHEMBL21040482 0.67 SMN1; SMN2 (0.48) ALDH1A1NPSR1
SCHEMBL19785990 0.66 BCHE (0.70) BCHEACHEKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0729465-B1 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE DAVIS & CO (US) 2003-01-22 EP disclosed
US-6005103-A TREATMENT OF BACTERIAL AND VIRAL INFECTIONS AND DISEASES, INCLUDING AIDS WARNER-LAMBERT COMPANY (US) 1999-12-21 US disclosed
EP-0729465-A1 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1996-09-04 EP disclosed
EP-0729466-A1 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1996-09-04 EP disclosed
WO-1995014013-A1 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1995-05-26 WO disclosed
WO-1995014014-A2 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1995-05-26 WO disclosed