SCHEMBL6955265

SCHEMBL6955265

Cc1cc(NC(=O)Oc2ccccc2)c(N2CCN(C(=O)OC(C)(C)C)CC2)nc1C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 2/20 0.48
KIT P10721 1/20 0.46
CKS1B P61024 2/20 0.44
SKP1 P63208 2/20 0.44
SKP2 Q13309 2/20 0.44
PTPN11 Q06124 1/20 0.44
ACHE P22303 1/20 0.43
BACE1 P56817 2/20 0.43
SMO Q99835 1/20 0.43
TLR9 Q9NR96 4/20 0.42
TLR7 Q9NYK1 2/20 0.41
NAMPT P43490 1/20 0.41
CCNK O75909 1/20 0.41
CCNA2 P20248 1/20 0.41
CDK2 P24941 1/20 0.41
CCND3 P30281 1/20 0.41
CDK9 P50750 1/20 0.41
CDK6 Q00534 1/20 0.41
P2RX7 Q99572 1/20 0.41
JAK2 O60674 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6964672 0.90 KIT (0.44) GBA1KITCKS1BSKP1SKP2
SCHEMBL6965424 0.83 SMO (0.42) SMO
SCHEMBL6942726 0.80 ALDH1A1 (0.49) CKS1BSKP1SKP2PTPN11BACE1
SCHEMBL6966613 0.79 KMT2A (0.45) TLR9NAMPTP2RX7
SCHEMBL6956575 0.78 MEN1 (0.45) GBA1KITTLR9NAMPTCCNK
SCHEMBL2366187 0.78 GBA1 (0.47) GBA1KITCKS1BSKP1SKP2
SCHEMBL6942730 0.75 GAA (0.69) PTPN11NAMPTJAK2JAK3
SCHEMBL8700308 0.75 PTPN11 (0.48) GBA1KITCKS1BSKP1SKP2
SCHEMBL14598720 0.74 GBA1 (0.47) GBA1KITCKS1BSKP1SKP2
SCHEMBL952359 0.72 GAA (0.60) CKS1BSKP1SKP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850222-B1 PIPERAZINE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF SAMJIN PHARM CO LTD (KR) 2003-05-28 EP disclosed
US-6028195-A AN ANTITUMOR AGENT WITH VERY LOW TOXICITIES SAMJIN PHARMACEUTICAL CO., LTD. (KR) 2000-02-22 US disclosed