SCHEMBL6955384

SCHEMBL6955384

COc1cccc2c(OC(C)=O)cc(C(=O)O)cc12

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.59
KDM4E B2RXH2 4/20 0.51
ALDH1A1 P00352 4/20 0.51
GAA P10253 1/20 0.51
RAB9A P51151 1/20 0.51
PKM P14618 3/20 0.51
HPGD P15428 3/20 0.51
HTT P42858 3/20 0.51
MAPK1 P28482 2/20 0.51
TTR P02766 2/20 0.51
MEN1 O00255 1/20 0.51
ABCC4 O15439 1/20 0.51
USP2 O75604 1/20 0.51
LMNA P02545 1/20 0.51
TP53 P04637 1/20 0.51
HSP90AA1 P07900 1/20 0.51
CHRM2 P08172 1/20 0.51
HSP90AB1 P08238 1/20 0.51
HTR1A P08908 1/20 0.51
ADRA2A P08913 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1812029 0.89 CA12 (0.55) TSHRKDM4EALDH1A1GAAPKM
SCHEMBL6042081 0.82 CDC25B (0.52) TSHRKDM4EALDH1A1GAARAB9A
SCHEMBL11207630 0.82 ESR1 (0.53) TSHRKDM4EALDH1A1GAAHPGD
SCHEMBL6959377 0.80 PTGS2 (0.57) KDM4EALDH1A1GAAPKMHPGD
SCHEMBL1812865 0.79 MRGPRX4 (0.51) TSHRKDM4EALDH1A1PKMHPGD
SCHEMBL6950752 0.78 MRGPRX4 (0.50) TSHRKDM4EALDH1A1RAB9APKM
SCHEMBL27562122 0.77 CYP3A4 (0.45) KDM4EALDH1A1RAB9AHPGDHTT
SCHEMBL4961779 0.77 ALDH1A1 (0.56) TSHRKDM4EALDH1A1GAARAB9A
SCHEMBL28857298 0.77 CA1 (0.69) TSHRKDM4ERAB9APKMHPGD
SCHEMBL7789471 0.76 SMN1; SMN2 (0.48) TSHRKDM4ERAB9APKMHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863875-B1 NEW 4-(OXYALKOXYPHENYL)-3-OXY-PIPERIDINES FOR TREATING HEART AND KIDNEY INSUFFICIENCY HOFFMANN LA ROCHE (CH) 2003-06-04 EP disclosed
EP-0863875-A1 NEW 4-(OXYALKOXYPHENYL)-3-OXY-PIPERIDINES FOR TREATING HEART AND KIDNEY INSUFFICIENCY F. HOFFMANN-LA ROCHE AG (CH) 1998-09-16 EP disclosed
WO-1997009311-A1 NEW 4-(OXYALKOXYPHENYL)-3-OXY-PIPERIDINES FOR TREATING HEART AND KIDNEY INSUFFICIENCY F. HOFFMANN-LA ROCHE AG (CH) 1997-03-13 WO disclosed