SCHEMBL6957549

SCHEMBL6957549

Nc1ccc(N(C=O)N(c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.52
ALDH1A1 P00352 5/20 0.52
TDP1 Q9NUW8 4/20 0.52
MAPT P10636 4/20 0.52
L3MBTL1 Q9Y468 4/20 0.52
CYP1A2 P05177 2/20 0.52
CYP2C9 P11712 2/20 0.52
CYP2C19 P33261 2/20 0.52
KDM4E B2RXH2 1/20 0.52
CYP2D6 P10635 1/20 0.52
MAOA P21397 4/20 0.38
MAOB P27338 4/20 0.38
CYP19A1 P11511 1/20 0.38
TSHR P16473 2/20 0.37
TAAR1 Q96RJ0 1/20 0.37
HSD17B10 Q99714 1/20 0.37
MAPK1 P28482 2/20 0.35
TP53 P04637 1/20 0.35
ALOX15 P16050 1/20 0.35
HTT P42858 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7593557 0.88 ALDH1A1 (0.37) CYP3A4ALDH1A1TDP1MAPTL3MBTL1
SCHEMBL9699565 0.78 CYP3A4 (0.58) CYP3A4ALDH1A1TDP1MAPTL3MBTL1
SCHEMBL7410822 0.74 ALDH1A1 (0.50) CYP3A4ALDH1A1TDP1MAPTL3MBTL1
SCHEMBL8862539 0.73 CYP3A4 (0.64) CYP3A4ALDH1A1TDP1MAPTL3MBTL1
Benzene SCHEMBL28589541 0.73 CYP3A4 (0.50) CYP3A4ALDH1A1TDP1MAPTL3MBTL1
SCHEMBL22733783 0.69 CYP3A4 (1.00) CYP3A4ALDH1A1TDP1MAPTL3MBTL1
SCHEMBL21311961 0.69 CYP3A4 (1.00) CYP3A4ALDH1A1TDP1MAPTL3MBTL1
SCHEMBL21538632 0.69 CYP3A4 (1.00) CYP3A4ALDH1A1TDP1MAPTL3MBTL1
Benzene SCHEMBL1030385 0.69 CYP3A4 (1.00) CYP3A4ALDH1A1TDP1MAPTL3MBTL1
SCHEMBL39413 0.69 CYP3A4 (1.00) CYP3A4ALDH1A1TDP1MAPTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0713483-B1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRAZENECA AB (SE) 2003-01-15 EP disclosed
US-6030985-A Amidine derivatives with nitric oxide synthetase activities ASTRA AKTIEBOLAG (SE) 2000-02-29 US disclosed
EP-0713483-A1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES Astra Aktiebolag (SE) 1996-05-29 EP disclosed
WO-1995005363-A1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRA AKTIEBOLAG (SE) 1995-02-23 WO disclosed