SCHEMBL9699565

SCHEMBL9699565

Nc1ccc(N(C=O)c2ccccc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.58
MAPT P10636 5/20 0.58
TDP1 Q9NUW8 4/20 0.58
ALDH1A1 P00352 4/20 0.58
L3MBTL1 Q9Y468 3/20 0.58
CYP1A2 P05177 2/20 0.58
CYP2C9 P11712 2/20 0.58
CYP2C19 P33261 2/20 0.58
KDM4E B2RXH2 1/20 0.58
CYP2D6 P10635 1/20 0.58
TSHR P16473 2/20 0.42
MAOA P21397 4/20 0.41
MAOB P27338 4/20 0.41
CYP19A1 P11511 1/20 0.41
TAAR1 Q96RJ0 1/20 0.41
HSD17B10 Q99714 1/20 0.41
MAPK1 P28482 2/20 0.39
TP53 P04637 1/20 0.39
ALOX15 P16050 1/20 0.39
HTT P42858 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13392612 0.91 ALDH1A1 (0.46) CYP3A4MAPTTDP1ALDH1A1L3MBTL1
SCHEMBL43388 0.86 ALDH1A1 (0.42) CYP3A4MAPTTDP1ALDH1A1L3MBTL1
SCHEMBL5516786 0.86 ALDH1A1 (0.42) CYP3A4MAPTTDP1ALDH1A1L3MBTL1
SCHEMBL823046 0.80 ALDH1A1 (0.39) CYP3A4MAPTTDP1ALDH1A1L3MBTL1
SCHEMBL28869065 0.78 TSHR (0.42) MAPTALDH1A1L3MBTL1CYP1A2KDM4E
SCHEMBL172583 0.78 CA12 (0.44) MAPTALDH1A1CYP2C19TSHRHTT
SCHEMBL6957549 0.78 CYP3A4 (0.52) CYP3A4MAPTTDP1ALDH1A1L3MBTL1
Benzene SCHEMBL28589541 0.77 CYP3A4 (0.50) CYP3A4MAPTTDP1ALDH1A1L3MBTL1
SCHEMBL10012838 0.77 ALDH1A1 (0.43) CYP3A4MAPTTDP1ALDH1A1CYP1A2
SCHEMBL10647182 0.75 CALM1 (0.48) CYP3A4TDP1ALDH1A1CYP2C9TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9067955-B2 Copper-catalyzed formation of carbon-heteroatom and carbon—carbon bonds MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2015-06-30 US disclosed
US-5114975-A Insecticides and miticides CIBA-GEIGY CORPORATION (US) 1992-05-19 US disclosed
EP-0304402-B1 ANILINOPHENYL THIOUREAS, ISOTHIOUREAS AND CARBODIIMIDES, THEIR PREPARATION AND THEIR USE IN PEST-CONTROL CIBA-GEIGY AG (CH) 1992-05-06 EP disclosed
US-5026730-A Anilinophenylthioureas, compositions containing them, and the use thereof in pest control CIBA-GEIGY CORPORATION (US) 1991-06-25 US disclosed
EP-0304402-A2 Anilinophenyl thioureas, isothioureas and carbodiimides, their preparation and their use in pest-control CIBA-GEIGY AG (CH) 1989-02-22 EP disclosed