SCHEMBL6957899

SCHEMBL6957899

COc1c(N2CC3CC3(N)C2)c(F)c(N)c2c(=O)c(C(=O)O)cn([C@@H]3C[C@@H]3F)c12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.51
KCNH2 Q12809 4/20 0.45
POLB P06746 2/20 0.45
CACNA1F O60840 1/20 0.45
MAPK1 P28482 1/20 0.45
CACNA1D Q01668 1/20 0.45
CACNA1S Q13698 1/20 0.45
CACNA1C Q13936 1/20 0.45
GSK3B P49841 10/20 0.42
TOP2A P11388 1/20 0.37
TOP2B Q02880 1/20 0.37
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
HPGD P15428 2/20 0.36
HSD17B10 Q99714 2/20 0.36
PRKD3 O94806 1/20 0.36
ALOX15 P16050 1/20 0.36
OPRM1 P35372 1/20 0.36
CLK2 P49760 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6973262 0.92 CACNA1F (0.53) CYP3A4KCNH2POLBCACNA1FMAPK1
SCHEMBL5787321 0.85 CYP3A4 (0.51) CYP3A4KCNH2POLBCACNA1FMAPK1
SCHEMBL5787325 0.85 CYP3A4 (0.51) CYP3A4KCNH2POLBCACNA1FMAPK1
SCHEMBL6957895 0.85 KCNH2 (0.42) CYP3A4KCNH2POLBCACNA1FMAPK1
SCHEMBL6948985 0.84 CYP3A4 (0.58) CYP3A4KCNH2POLBKDM4EALDH1A1
SCHEMBL6975592 0.81 CACNA1F (0.40) CYP3A4KCNH2POLBCACNA1FMAPK1
SCHEMBL502617 0.81 GSK3B (0.51) CYP3A4KCNH2POLBCACNA1FMAPK1
SCHEMBL5783269 0.81 GSK3B (0.51) CYP3A4KCNH2POLBCACNA1FMAPK1
SCHEMBL4671496 0.81 CACNA1F (0.57) CYP3A4KCNH2POLBCACNA1FMAPK1
SCHEMBL6163513 0.80 CYP3A4 (0.50) CYP3A4KCNH2POLBCACNA1FMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1304329-A2 Pyridonecarboxylic acid derivatives and their use as antibacterial agents DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2003-04-23 EP disclosed
EP-0807630-A1 HETEROCYCLIC COMPOUNDS DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1997-11-19 EP disclosed