SCHEMBL695795

SCHEMBL695795

N#CC1(NC(=O)[C@@H]2C[C@@H](S(=O)(=O)c3ccc(F)cc3C(F)(F)F)CN2)CC1

nearest known ligand 0.78

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CTSS P25774 19/20 0.78
CTSC P53634 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL694322 0.90 CTSS (0.77) CTSSCTSC
Hydrochloric Acid SCHEMBL695437 0.89 CTSS (0.75) CTSSCTSC
SCHEMBL695316 0.89 CTSS (0.66) CTSSCTSC
Hydrochloric Acid SCHEMBL696606 0.88 CTSS (0.65) CTSSCTSC
SCHEMBL696004 0.88 CTSS (1.00) CTSSCTSC
SCHEMBL695956 0.88 CTSS (1.00) CTSSCTSC
SCHEMBL696446 0.87 CTSS (0.64) CTSSCTSC
Hydrochloric Acid SCHEMBL695373 0.87 CTSS (0.98) CTSSCTSC
SCHEMBL696453 0.86 CTSS (0.71) CTSS
SCHEMBL2108232 0.85 CTSS (0.69) CTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8163793-B2 Proline derivatives HOFFMAN-LA ROCHE INC. (US) 2012-04-24 US disclosed
EP-2421826-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. Hoffmann-La Roche AG (CH) 2012-02-29 EP disclosed
WO-2010121918-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2010-10-28 WO disclosed