SCHEMBL6958605

SCHEMBL6958605

C(=C/c1ccc2ccccc2c1)\Cc1c[nH]cn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RELA Q04206 1/20 0.44
PTGS1 P23219 1/20 0.40
NQO2 P16083 2/20 0.38
ALDH1A1 P00352 2/20 0.38
GLA P06280 1/20 0.38
MAPT P10636 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
GRIK1 P39086 1/20 0.37
GRIK2 Q13002 1/20 0.37
GRIK3 Q13003 1/20 0.37
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
CHRNA7 P36544 1/20 0.36
KDM4E B2RXH2 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
PTPN1 P18031 1/20 0.34
CYP1A1 P04798 1/20 0.34
CYP1A2 P05177 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6958610 1.00 RELA (0.44) RELAPTGS1NQO2ALDH1A1GLA
SCHEMBL9519041 0.82 RAB9A (0.39) SMN1; SMN2KDM4EL3MBTL1CYP1A2CYP3A4
SCHEMBL28260827 0.72 RELA (0.55) RELAPTGS1NQO2ALDH1A1GLA
SCHEMBL2355562 0.72 RELA (0.55) RELAPTGS1NQO2ALDH1A1GLA
SCHEMBL2103758 0.71 BACE1 (0.47) CYP1A2CYP2D6
SCHEMBL7974933 0.71 TDP1 (0.51) ALDH1A1MAPTSMN1; SMN2KDM4E
SCHEMBL7362771 0.70 BACE1 (0.48) CYP1A2CYP2D6
SCHEMBL224386 0.69 ANPEP (0.39) MAPTL3MBTL1
SCHEMBL5050698 0.68 RELA (0.86) RELAPTGS1NQO2ALDH1A1GLA
SCHEMBL5552162 0.68 RELA (0.86) RELAPTGS1NQO2ALDH1A1GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0974584-B1 FUSED RING COMPOUNDS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-01-15 EP disclosed
US-6420375-B1 ANTITUMOR TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-07-16 US disclosed
EP-0974584-A1 FUSED RING COMPOUNDS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2000-01-26 EP disclosed