SCHEMBL6958634

SCHEMBL6958634

N=C(Nc1ccc(CCOC(=O)Nc2ccccc2)cc1)c1cccs1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 9/20 0.52
RAB9A P51151 9/20 0.52
SMN1; SMN2 Q16637 4/20 0.52
RECQL P46063 1/20 0.52
MGLL Q99685 1/20 0.50
ROCK2 O75116 1/20 0.47
TSHR P16473 1/20 0.47
MEN1 O00255 6/20 0.46
KMT2A Q03164 6/20 0.46
TP53 P04637 3/20 0.46
ALDH1A1 P00352 1/20 0.46
KDM4E B2RXH2 1/20 0.44
LMNA P02545 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
CHRNA7 P36544 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6958640 0.80 NOS1 (0.52) NPC1RAB9ASMN1; SMN2RECQLMGLL
SCHEMBL9038704 0.80 NPC1 (0.55) NPC1RAB9ASMN1; SMN2ROCK2MEN1
SCHEMBL6962657 0.80 TRPV1 (0.55) NPC1RAB9ASMN1; SMN2MEN1KMT2A
Iodide SCHEMBL6962649 0.79 NPC1 (0.54) NPC1RAB9ASMN1; SMN2ROCK2MEN1
SCHEMBL7081200 0.78 NPC1 (0.56) NPC1RAB9ASMN1; SMN2TSHRMEN1
Phenethyl Phenylcarbamate SCHEMBL1835027 0.78 NPC1 (0.81) NPC1RAB9ASMN1; SMN2RECQLMGLL
SCHEMBL6280367 0.78 RAB9A (0.53) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL9037372 0.78 NPC1 (0.51) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL4627573 0.77 NPC1 (0.52) NPC1RAB9ASMN1; SMN2ROCK2MEN1
SCHEMBL4627215 0.77 TRPV1 (0.52) NPC1RAB9ASMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995005363-A1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRA AKTIEBOLAG (SE) 1995-02-23 WO claimed
EP-0713483-B1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRAZENECA AB (SE) 2003-01-15 EP disclosed
US-6030985-A Amidine derivatives with nitric oxide synthetase activities ASTRA AKTIEBOLAG (SE) 2000-02-29 US disclosed
US-5807885-A Amidine derivatives with nitric oxide synthetase activities ASTRA AKTIEBOLAG (SE) 1998-09-15 US disclosed