SCHEMBL6958799

SCHEMBL6958799

COc1cccc(CCNC(=S)Nc2nc(-c3cccnc3)cs2)c1

nearest known ligand 0.72

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.72
CYP3A4 P08684 10/20 0.59
ROCK1 Q13464 8/20 0.59
MAPT P10636 3/20 0.59
PRKACA P17612 2/20 0.59
NPC1 O15118 4/20 0.58
RAB9A P51151 4/20 0.58
MEN1 O00255 2/20 0.58
KMT2A Q03164 2/20 0.58
ROCK2 O75116 2/20 0.58
SMN1; SMN2 Q16637 3/20 0.56
CYP1A2 P05177 1/20 0.56
CYP2D6 P10635 1/20 0.56
CYP2C9 P11712 1/20 0.56
CYP2C19 P33261 1/20 0.56
ALDH1A1 P00352 2/20 0.52
HPGD P15428 1/20 0.52
HSD17B10 Q99714 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6959245 0.90 MAPT (0.71) HTTCYP3A4ROCK1MAPTNPC1
SCHEMBL6962797 0.88 ROCK2 (0.56) HTTCYP3A4ROCK1MAPTNPC1
SCHEMBL6962350 0.86 ROCK1 (0.57) HTTCYP3A4ROCK1MAPTPRKACA
SCHEMBL6953866 0.86 MEN1 (0.56) HTTCYP3A4ROCK1MAPTNPC1
SCHEMBL6956316 0.86 MAPT (0.58) HTTCYP3A4ROCK1MAPTPRKACA
SCHEMBL6964598 0.86 NPC1 (0.59) HTTCYP3A4ROCK1MAPTPRKACA
SCHEMBL6962738 0.85 ALDH1A1 (0.70) HTTROCK1MAPTPRKACANPC1
SCHEMBL6956968 0.85 MAPT (0.55) HTTCYP3A4ROCK1MAPTNPC1
SCHEMBL6956833 0.85 MAPT (0.56) HTTCYP3A4ROCK1MAPTPRKACA
SCHEMBL6958055 0.84 MEN1 (0.65) HTTCYP3A4ROCK1MAPTPRKACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0540143-B1 Compounds and methods for inhibition of HIV and related viruses MEDIVIR AB (SE) 2003-02-05 EP disclosed
US-5658907-A THIOUREA VIRICIDES MEDIVIR A/B (SE) 1997-08-19 US disclosed
US-5593993-A VIRICIDES FOR HTLV TREATMENT OF AIDS MEDIVIR AB (SE) 1997-01-14 US disclosed
EP-0540143-A2 Compounds and methods for inhibition of HIV and related viruses Medivir Aktiebolag (SE) 1993-05-05 EP disclosed
WO-1993003022-A1 COMPOUNDS AND METHODS FOR INHIBITION OF HIV AND RELATED VIRUSES MEDIVIR AB (SE) 1993-02-18 WO disclosed