SCHEMBL6959025

SCHEMBL6959025

N#Cc1ccc2cc(CCCC(=O)N3CCCC(Cc4ccccc4)C3)[nH]c2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.44
DRD4 P21917 2/20 0.44
DRD3 P35462 2/20 0.44
HTR2A P28223 1/20 0.43
CCR3 P51677 1/20 0.43
TNKS O95271 1/20 0.42
PARP1 P09874 1/20 0.42
PARP2 Q9UGN5 1/20 0.42
KDM4E B2RXH2 1/20 0.42
MAPK1 P28482 1/20 0.42
TACR3 P29371 2/20 0.41
MGLL Q99685 1/20 0.41
GRIN2D O15399 1/20 0.41
GRIN3B O60391 1/20 0.41
GRIN1 Q05586 1/20 0.41
GRIN2A Q12879 1/20 0.41
GRIN2B Q13224 1/20 0.41
GRIN2C Q14957 1/20 0.41
GRIN3A Q8TCU5 1/20 0.41
CHRNB2 P17787 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6953902 0.93 DRD2 (0.44) DRD2DRD4DRD3HTR2ACCR3
SCHEMBL6956012 0.87 TACR3 (0.43) TNKSPARP1PARP2KDM4EMAPK1
SCHEMBL6958696 0.87 MEN1 (0.46) TNKSPARP1PARP2KDM4EMAPK1
SCHEMBL6953001 0.85 MEN1 (0.56) HTR2ACCR3KDM4EMEN1NPC1
SCHEMBL6949095 0.83 MEN1 (0.47) KDM4EMAPK1TACR3GRIN2DGRIN3B
SCHEMBL6955497 0.82 CCR3 (0.51) DRD2DRD4DRD3HTR2ACCR3
SCHEMBL6952765 0.82 TACR1 (0.52) HTR2ACCR3TACR3TACR1KMT2A
SCHEMBL18782564 0.82 AKR1C3 (0.50) TACR3GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL6954412 0.82 TACR3 (0.43) KDM4EMAPK1TACR3GRIN2DGRIN3B
SCHEMBL6958058 0.82 MEN1 (0.55) TNKSPARP1PARP2KDM4EMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0993458-B1 3-BENZYLPIPERIDINE MERCK PATENT GMBH (DE) 2003-04-09 EP disclosed
EP-0993458-A1 3-BENZYLPIPERIDINE MERCK PATENT GmbH (DE) 2000-04-19 EP disclosed
WO-1998057953-A1 3-BENZYLPIPERIDINE MERCK PATENT GMBH (DE) 1998-12-23 WO disclosed